In vitro interactions between piperaquine, dihydroartemisinin, and other conventional and novel antimalarial drugs

Antimicrob Agents Chemother. 2006 Aug;50(8):2883-5. doi: 10.1128/AAC.00177-06.

Abstract

In an in vitro assessment of antimalarial combinations, dihydroartemisinin (DHA) showed no interaction or was mildly antagonistic when combined with piperaquine, pyronaridine, or naphthoquine. Interactions between 4-aminoquinolines and related drugs were also indifferent/antagonistic. The clinical significance of mildly antagonistic DHA combinations is uncertain but may become important if parasite drug sensitivity declines.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antimalarials / pharmacology*
  • Artemisinins / pharmacology*
  • Drug Combinations
  • Drug Interactions
  • In Vitro Techniques
  • Plasmodium falciparum / drug effects
  • Plasmodium falciparum / genetics
  • Plasmodium falciparum / growth & development
  • Quinolines / pharmacology*

Substances

  • Antimalarials
  • Artemisinins
  • Drug Combinations
  • Quinolines
  • piperaquine