Dominant-negative E-cadherin inhibits the invasiveness of inflammatory breast cancer cells in vitro

J Cancer Res Clin Oncol. 2007 Feb;133(2):83-92. doi: 10.1007/s00432-006-0140-6. Epub 2006 Aug 24.

Abstract

E-cadherin is a transmembrane glycoprotein which mediates epithelial cell-to-cell adhesion function as a tumor suppressor and frequently loss of expression in a wide spectrum of human cancer. However, recent studies demonstrated that E-cadherin was always over-expressed in inflammatory breast cancer (IBC) specimen and cell lines, which is a clinical extreme malignancy of breast cancer. It is hypothesized that the gain and not the loss of the E-cadherin axis contributes to the IBC unique phenotype. To test this assumption, we generated dominant negative mutant E-cadherin high-expression inflammatory breast cancer cells by introduced dominant negative mutant E-cadherin (H-2kd-E-cad) cDNA into human IBC SUM149 cells. Our studies demonstrated that the ability of invasion of SUM149 cells was significantly inhibited by H-2kd-E-cad via down-regulation of MMP-1 and MMP-9 expression. The underlying signal pathway of MAPK phosphorylated Erk 1/2(P44/42) in H-2kd-E-cad-transfected SUM149 cells was significantly down-regulated compared to parental and mock contrast. Our studies provided further functional evidence as the gain of E-cadherin expression dedicated to the IBC malignant phenotype and the blockage of MAPK/Erk activation maybe a promising therapeutic target.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Breast Neoplasms / genetics
  • Breast Neoplasms / metabolism
  • Breast Neoplasms / pathology*
  • Cadherins / genetics*
  • Cadherins / metabolism
  • DNA, Complementary
  • Down-Regulation
  • Extracellular Signal-Regulated MAP Kinases / metabolism
  • Female
  • Humans
  • Matrix Metalloproteinase 1 / genetics
  • Matrix Metalloproteinase 1 / metabolism
  • Matrix Metalloproteinase 9 / genetics
  • Matrix Metalloproteinase 9 / metabolism
  • Mutation
  • Neoplasm Invasiveness
  • Phenotype
  • Signal Transduction
  • Transfection
  • Tumor Cells, Cultured

Substances

  • Cadherins
  • DNA, Complementary
  • Extracellular Signal-Regulated MAP Kinases
  • Matrix Metalloproteinase 9
  • Matrix Metalloproteinase 1