Cytochrome P450-dependent arachidonic acid metabolites, 19- and 20-hydroxyeicosatetraenoic acids, enhance sodium-potassium ATPase activity in vascular smooth muscle

J Cardiovasc Pharmacol. 1990 Sep;16(3):438-43. doi: 10.1097/00005344-199009000-00013.

Abstract

Several cytochrome P450-dependent arachidonic acid metabolites have been shown to affect Na+,K(+)-ATPase activity. In the present study, we tested the effect of omega- and omega - 1-hydroxylated products, i.e., 19- and 20-hydroxyeicosatetraenoic acids (19- and 20-HETE), on the K-induced relaxation in rat aortic rings. 19-HETE and 20-HETE increased the magnitude of the potassium-induced relaxation in a dose-dependent fashion (10(-7)-10(-5) M). The inhibitory effect of ouabain on the potassium-induced relaxation was reversed by both 19- and 20-HETE. In addition, indomethacin fully inhibited the stimulatory effect of 19- and 20-HETE on relaxation induced by potassium. Vascular ouabain-sensitive 86Rb uptake was also increased by 19- and 20-HETE. These observations suggest that 19- and 20-HETE stimulate vascular Na+,K(+)-ATPase via their conversion by cyclooxygenase to prostaglandin-like material.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Analysis of Variance
  • Animals
  • Aorta, Thoracic
  • Cytochrome P-450 Enzyme System / physiology*
  • Hydroxyeicosatetraenoic Acids / pharmacology
  • Hydroxyeicosatetraenoic Acids / physiology*
  • In Vitro Techniques
  • Indomethacin / pharmacology
  • Male
  • Muscle Relaxation / drug effects
  • Muscle, Smooth, Vascular / enzymology*
  • Ouabain / pharmacology
  • Potassium / pharmacology
  • Rats
  • Rats, Inbred Strains
  • Rubidium Radioisotopes
  • Sodium-Potassium-Exchanging ATPase / metabolism*

Substances

  • Hydroxyeicosatetraenoic Acids
  • Rubidium Radioisotopes
  • Ouabain
  • 19-hydroxy-5,8,11,14-eicosatetraenoic acid
  • 20-hydroxy-5,8,11,14-eicosatetraenoic acid
  • Cytochrome P-450 Enzyme System
  • Sodium-Potassium-Exchanging ATPase
  • Potassium
  • Indomethacin