Failure of calcium microdomain generation and pathological consequences

Cell Calcium. 2006 Nov-Dec;40(5-6):593-600. doi: 10.1016/j.ceca.2006.08.020. Epub 2006 Oct 17.

Abstract

Normal physiological regulation depends on Ca(2+) microdomains, because there is a need to spatially separate Ca(2+) regulation of different cellular processes. It is only possible to generate local Ca(2+) signals transiently; so, there is an important functional link between Ca(2+) spiking and microdomains. The pancreatic acinar cell provides a useful cell biological model, because of its clear structural and functional polarization. Although local Ca(2+) spiking in the apical (granular) microdomain regulates fluid and enzyme secretion, prolonged global elevations of the cytosolic Ca(2+) concentration are associated with the human disease acute pancreatitis, in which proteases in the granular region become inappropriately activated and digest the pancreas and its surroundings. A major cause of pancreatitis is alcohol abuse and it has now been established that fatty acid ethyl esters and fatty acids, non-oxidative alcohol metabolites, are principally responsible for causing the acinar cell damage. The fatty acid ethyl esters release Ca(2+) from the endoplasmic reticulum and the fatty acids inhibit markedly mitochondrial ATP generation, which prevents the acinar cell from disposing of the excess Ca(2+) in the cytosol. Because of the abolition of ATP-dependent Ca(2+) pump activity, all intracellular Ca(2+) concentration gradients disappear and the most important part of the normal regulatory machinery is thereby destroyed. The end stage is necrosis.

Publication types

  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Adenosine Triphosphate / metabolism
  • Animals
  • Calcium Signaling* / physiology
  • Cytosol / metabolism
  • Endoplasmic Reticulum / physiology
  • Epithelial Cells / physiology
  • Esters / metabolism
  • Fatty Acids / metabolism
  • Homeostasis
  • Inositol 1,4,5-Trisphosphate Receptors / physiology
  • Membrane Microdomains* / physiology
  • Models, Biological
  • Pancreas / cytology
  • Pancreatitis / physiopathology*
  • Ryanodine Receptor Calcium Release Channel / physiology

Substances

  • Esters
  • Fatty Acids
  • Inositol 1,4,5-Trisphosphate Receptors
  • Ryanodine Receptor Calcium Release Channel
  • Adenosine Triphosphate