Rapamycin is efficacious against primary effusion lymphoma (PEL) cell lines in vivo by inhibiting autocrine signaling

Blood. 2007 Mar 1;109(5):2165-73. doi: 10.1182/blood-2006-06-028092. Epub 2006 Nov 2.

Abstract

The antitumor potency of the mTOR inhibitor rapamycin (sirolimus) is the subject of intense investigations. Primary effusion lymphoma (PEL) appears as an AIDS-defining lymphoma and like Kaposi sarcoma has been linked to Kaposi sarcoma-associated herpesvirus (KSHV). We find that (1) rapamycin is efficacious against PEL in culture and in a murine xenograft model; (2) mTOR, its activator Akt, and its target p70S6 kinase are phosphorylated in PEL; (3) rapamycin inhibits mTOR signaling as determined by S6 phosphorylation; (4) KSHV transcription is unaffected; (5) inhibition of IL-10 signaling correlates with drug sensitivity; and (6) addition of exogenous IL-10 or IL-6 can reverse the rapamycin growth arrest. This validates sirolimus as a new treatment option for PEL.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Autocrine Communication / drug effects*
  • Cell Line, Tumor
  • Cell Proliferation / drug effects
  • Cytokines / biosynthesis
  • Cytokines / genetics
  • Disease Progression
  • Herpesvirus 8, Human / drug effects
  • Herpesvirus 8, Human / genetics
  • Humans
  • Lymphoma / metabolism*
  • Lymphoma / pathology*
  • Mice
  • RNA, Messenger / genetics
  • Sirolimus / pharmacology*
  • Transcription, Genetic / genetics
  • Xenograft Model Antitumor Assays

Substances

  • Cytokines
  • RNA, Messenger
  • Sirolimus