Third activity of Bordetella adenylate cyclase (AC) toxin-hemolysin. Membrane translocation of AC domain polypeptide promotes calcium influx into CD11b+ monocytes independently of the catalytic and hemolytic activities

J Biol Chem. 2007 Feb 2;282(5):2808-20. doi: 10.1074/jbc.M609979200. Epub 2006 Dec 4.

Abstract

The Bordetella adenylate cyclase toxin-hemolysin (CyaA) targets phagocytes expressing the alpha(M)beta2 integrin (CD11b/CD18), permeabilizes their membranes by forming small cation-selective pores, and delivers into cells a calmodulin-activated adenylate cyclase (AC) enzyme that dissipates cytosolic ATP into cAMP. We describe here a third activity of CyaA that yields elevation of cytosolic calcium concentration ([Ca2+]i) in target cells. The CyaA-mediated [Ca2+]i increase in CD11b+ J774A.1 monocytes was inhibited by extracellular La3+ ions but not by nifedipine, SK&F 96365, flunarizine, 2-aminoethyl diphenylborinate, or thapsigargin, suggesting that influx of Ca2+ into cells was not because of receptor signaling or opening of conventional calcium channels by cAMP. Compared with intact CyaA, a CyaA-AC- toxoid unable to generate cAMP promoted a faster, albeit transient, elevation of [Ca2+]i. This was not because of cell permeabilization by the CyaA hemolysin pores, because a mutant exhibiting a strongly enhanced pore-forming activity (CyaA-E509K/E516K), but unable to deliver the AC domain into cells, was also unable to elicit a [Ca2+]i increase. Further mutations interfering with AC translocation into cells, such as proline substitutions of glutamate residues 509 or 570 or deletion of the AC domain as such, reduced or ablated the [Ca2+]i-elevating capacity of CyaA. Moreover, structural alterations within the AC domain, because of insertion of various oligopeptides, differently modulated the kinetics and extent of Ca2+ influx elicited by the respective AC- toxoids. Hence, the translocating AC polypeptide itself appears to participate in formation of a novel type of membrane path for calcium ions, contributing to action of CyaA in an unexpected manner.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adenosine Triphosphate / metabolism
  • Adenylate Cyclase Toxin / chemistry
  • Adenylate Cyclase Toxin / genetics
  • Adenylate Cyclase Toxin / isolation & purification
  • Adenylate Cyclase Toxin / metabolism*
  • Adenylyl Cyclases / metabolism*
  • Amino Acid Substitution
  • Animals
  • Biological Transport
  • CD11b Antigen / physiology*
  • Calcium / metabolism*
  • Catalysis
  • Cell Line
  • Cell Membrane / physiology
  • Cyclic AMP / metabolism
  • Hemolysis
  • Macrophages / physiology
  • Mice
  • Monocytes / physiology*
  • Mutagenesis, Site-Directed
  • Polymerase Chain Reaction
  • Recombinant Proteins / chemistry
  • Recombinant Proteins / isolation & purification
  • Recombinant Proteins / metabolism
  • Sheep

Substances

  • Adenylate Cyclase Toxin
  • CD11b Antigen
  • Recombinant Proteins
  • Adenosine Triphosphate
  • Cyclic AMP
  • Adenylyl Cyclases
  • Calcium