Liver X receptors regulate dendritic cell phenotype and function through blocked induction of the actin-bundling protein fascin

Blood. 2007 May 15;109(10):4288-95. doi: 10.1182/blood-2006-08-043422. Epub 2007 Jan 25.

Abstract

Liver X receptors (LXRs) are nuclear receptors regulating lipid and cholesterol metabolism. Recent data revealed a cross talk between LXR and Toll-like receptor signaling in macrophages, indicating a role in immunity. Here, we show that LXRalpha is expressed in human myeloid dendritic cells (DCs) and induced during differentiation of monocyte-derived DCs, whereas LXRbeta is expressed constitutively at a very low level. LXR activation by 2 different LXR agonists strongly interfered with lipopolysaccharide (LPS)-induced but not with CD40L-induced DC maturation by altering DC morphology and suppressing interleukin-12-but enhancing interleukin-10-secretion. LXR activation in DCs largely blocked their T-cell stimulatory ability despite essentially unaltered expression of various antigen-presenting and costimulatory molecules. Immunologic synapse formation was significantly inhibited by LXR activation along with a complete block in LPS- but not CD40L-induced expression of the actin-bundling protein fascin. Notably, overexpression of fascin in LXR agonist-treated DCs restored immunologic synapse formation and restored their ability to activate T cells. In conclusion, our data reveal LXR as a potent modulator of DC maturation and function mediated in part by blocking the expression of fascin. Due to the central position of DCs in immunity, LXRalpha could be a potential novel target for immunomodulation.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Carrier Proteins / genetics*
  • Carrier Proteins / metabolism
  • Cells, Cultured
  • DNA-Binding Proteins / agonists
  • DNA-Binding Proteins / metabolism
  • DNA-Binding Proteins / physiology*
  • Dendritic Cells / cytology*
  • Dendritic Cells / drug effects
  • Dendritic Cells / physiology*
  • Female
  • Gene Expression Regulation / drug effects
  • Humans
  • Hydrocarbons, Fluorinated
  • Liver X Receptors
  • Male
  • Microfilament Proteins / genetics*
  • Microfilament Proteins / metabolism
  • Orphan Nuclear Receptors
  • Phenotype*
  • Receptors, Cytoplasmic and Nuclear / agonists
  • Receptors, Cytoplasmic and Nuclear / metabolism
  • Receptors, Cytoplasmic and Nuclear / physiology*
  • Sulfonamides / pharmacology
  • Transfection

Substances

  • Carrier Proteins
  • DNA-Binding Proteins
  • Hydrocarbons, Fluorinated
  • Liver X Receptors
  • Microfilament Proteins
  • NR1H3 protein, human
  • Orphan Nuclear Receptors
  • Receptors, Cytoplasmic and Nuclear
  • Sulfonamides
  • T0901317
  • fascin