Targeting of the transcription factor STAT4 by antisense phosphorothioate oligonucleotides suppresses collagen-induced arthritis

J Immunol. 2007 Mar 15;178(6):3427-36. doi: 10.4049/jimmunol.178.6.3427.

Abstract

The transcription factor STAT4 mediates signals of various proinflammatory cytokines, such as IL-12, IL-15, and IL-23, that initiate and stabilize Th1 cytokine production. Although Th1 cytokine production has been suggested to play a major pathogenic role in rheumatoid arthritis, the role of STAT4 in this disease is poorly understood. In this study, we demonstrate a key functional role of STAT4 in murine collagen-induced arthritis (CIA). In initial studies we found that STAT4 expression is strongly induced in CD4(+) T cells and to a lesser extent in CD11b(+) APCs during CIA. To analyze the role of STAT4 for arthritis manifestation, we next investigated the outcome of interfering with STAT4 gene expression in CIA by using STAT4-deficient mice. Interestingly, STAT4-deficient mice developed significantly less severe arthritis than wild-type control mice and the T cells from such mice produced less IL-6, TNF, and IL-17. In addition, the targeting of STAT4 expression by a specific antisense phosphorothioate oligonucleotide directed at the translation start site suppressed STAT4 levels and signs of CIA even when applied during the onset of disease manifestation. These data suggest a key regulatory role of STAT4 in the pathogenesis and manifestation of murine collagen-induced arthritis. Furthermore, the targeting of STAT4 emerges as a novel approach to therapy for chronic arthritis.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antigen-Presenting Cells / immunology
  • Antigen-Presenting Cells / pathology
  • Arthritis, Experimental / drug therapy
  • Arthritis, Experimental / immunology*
  • Arthritis, Experimental / pathology
  • Arthritis, Rheumatoid / drug therapy
  • Arthritis, Rheumatoid / immunology*
  • Arthritis, Rheumatoid / pathology
  • CD11b Antigen / immunology
  • Cells, Cultured
  • Codon, Initiator / antagonists & inhibitors
  • Codon, Initiator / immunology
  • Mice
  • Mice, Inbred BALB C
  • Mice, Knockout
  • Oligonucleotides, Antisense / pharmacology*
  • STAT4 Transcription Factor / antagonists & inhibitors*
  • STAT4 Transcription Factor / deficiency
  • STAT4 Transcription Factor / immunology
  • Th1 Cells / immunology*
  • Th1 Cells / pathology
  • Thionucleotides / pharmacology*

Substances

  • CD11b Antigen
  • Codon, Initiator
  • Oligonucleotides, Antisense
  • STAT4 Transcription Factor
  • Stat4 protein, mouse
  • Thionucleotides