Endogenous platelet factor 4 stimulates activated protein C generation in vivo and improves survival after thrombin or lipopolysaccharide challenge

Blood. 2007 Sep 15;110(6):1903-5. doi: 10.1182/blood-2007-03-081901. Epub 2007 May 31.

Abstract

Pharmacologic infusion of activated protein C (APC) improves survival in severe sepsis, and platelet factor 4 (PF4) accelerates APC generation in a primate thrombin-infusion model. We now tested whether endogenous platelet PF4 content affects APC generation. Mice completely deficient in PF4 (mPF4(-/-)) had impaired APC generation and survival after thrombin infusion, similar to the impairment seen in heterozygote protein C-deficient (PC(+/-)) mice. Transgenic mice overexpressing human PF4 (hPF4(+)) had increased plasma APC generation. Overexpression of platelet PF4 compensated for the defect seen in PC(+/-) mice. In both a thrombin and a lipopolysaccharide (LPS) survival model, hPF4(+) and PC(+/-)/hPF4(+) mice had improved survival. Further, infusion of hPF4(+) platelets improved survival of wild-type mice after an LPS challenge. These studies suggest that endogenous PF4 release may have biologic consequences for APC generation and survival in clinical sepsis. Infusions of PF4-rich platelets may be an effective strategy to improve outcome in this setting.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Animals
  • Anticoagulants / pharmacology
  • Blood Coagulation
  • Blood Platelets / drug effects
  • Blood Platelets / metabolism
  • Endotoxemia / metabolism
  • Endotoxemia / pathology
  • Endotoxemia / prevention & control*
  • Hemostatics / pharmacology*
  • Heterozygote
  • Humans
  • Lipopolysaccharides / pharmacology*
  • Mice
  • Mice, Knockout
  • Mice, Transgenic
  • Platelet Factor 4 / genetics
  • Platelet Factor 4 / physiology*
  • Protein C / biosynthesis*
  • Protein C Deficiency
  • Survival Rate
  • Thrombin / pharmacology*

Substances

  • Anticoagulants
  • Hemostatics
  • Lipopolysaccharides
  • Protein C
  • Platelet Factor 4
  • Thrombin