Association study between clinical response to rizatriptan and some candidate genes

J Headache Pain. 2007 Jun;8(3):185-9. doi: 10.1007/s10194-007-0388-5. Epub 2007 Jun 11.

Abstract

The aim of this study was to test genetic differences in the clinical response to rizatriptan in patients affected by migraine without aura. These genetic differences could be explained by various genes, the HTR1B, encoding the 5-HT(1) receptor subtype, MAOA gene that encodes the monoamino-oxidase, the main metabolic enzyme of this triptan, SLC6A4 (gene encoding the serotonin transporter) and DRD(2) (gene encoding the D(2) receptor), both involved in the pathogenesis of migraine. Fifty unrelated patients affected by migraine without aura (IHS) were included. Patients were divided into two groups (responders and non-responders) according to clinical response. Thirty-one out of fifty patients responded to rizatriptan. A significant difference among the two groups was observed in both allele (p=0.02) and genotype distribution (p=0.03) of DRD2/NcoI. The significant association with the DRD2/NcoI polymorphism in responders suggested that the DRD2/NcoI C allele may be considered a susceptibility factor heralding a good response to rizatriptan.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Alleles
  • Drug Resistance
  • Female
  • Genotype
  • Humans
  • Male
  • Middle Aged
  • Migraine without Aura / drug therapy*
  • Migraine without Aura / genetics*
  • Monoamine Oxidase / genetics
  • Polymorphism, Genetic
  • Prospective Studies
  • Receptor, Serotonin, 5-HT1B / genetics
  • Receptors, Dopamine D2 / genetics
  • Reverse Transcriptase Polymerase Chain Reaction
  • Serotonin Plasma Membrane Transport Proteins / genetics
  • Serotonin Receptor Agonists / therapeutic use*
  • Treatment Outcome
  • Triazoles / therapeutic use*
  • Tryptamines / therapeutic use*

Substances

  • HTR1B protein, human
  • Receptor, Serotonin, 5-HT1B
  • Receptors, Dopamine D2
  • Serotonin Plasma Membrane Transport Proteins
  • Serotonin Receptor Agonists
  • Triazoles
  • Tryptamines
  • rizatriptan
  • Monoamine Oxidase