FOXP1: a potential therapeutic target in cancer

Expert Opin Ther Targets. 2007 Jul;11(7):955-65. doi: 10.1517/14728222.11.7.955.

Abstract

Forkhead Box P1 (FOXP1) is a member of the FOX family of transcription factors which have a broad range of functions. Foxp1 is widely expressed and has been shown to have a role in cardiac, lung and lymphocyte development. FOXP1 is targeted by recurrent chromosome translocations and its overexpression confers a poor prognosis in a number of types of lymphomas, suggesting it may function as an oncogene. In contrast, FOXP1 localises to a tumour suppressor locus at 3p14.1 and loss of FOXP1 expression in breast cancer is associated with a worse outcome, suggesting FOXP1 may function as a tumour suppressor in other tissue types. These data suggest that FOXP1 may not only be useful in prognosis but also may be used to develop FOXP1-directed therapeutic strategies.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Review

MeSH terms

  • Animals
  • Forkhead Transcription Factors / genetics
  • Forkhead Transcription Factors / metabolism*
  • Humans
  • Neoplasms / genetics
  • Neoplasms / metabolism*
  • Oncogenes / genetics
  • Repressor Proteins / genetics
  • Repressor Proteins / metabolism*

Substances

  • FOXP1 protein, human
  • Forkhead Transcription Factors
  • Repressor Proteins