Inhibitory effect of PACAP-38 on acute neurogenic and non-neurogenic inflammatory processes in the rat

Peptides. 2007 Sep;28(9):1847-55. doi: 10.1016/j.peptides.2007.07.001. Epub 2007 Jul 7.

Abstract

Inhibitory actions of pituitary adenylate cyclase activating polypeptide (PACAP) have been described on cellular/vascular inflammatory components, but there are few data concerning its role in neurogenic inflammation. In this study we measured PACAP-like immunoreactivity with radioimmunoassay in the rat plasma and showed a two-fold elevation in response to systemic stimulation of capsaicin-sensitive sensory nerves by resiniferatoxin, but not after local excitation of cutaneous afferents. Neurogenic plasma extravasation in the plantar skin induced by intraplantar capsaicin or resiniferatoxin, as well as carrageenan-induced paw edema were significantly diminished by intraperitoneal PACAP-38. In summary, these results demonstrate that PACAP is released from activated capsaicin-sensitive afferents into the systemic circulation. It diminishes acute pure neurogenic and mixed-type inflammatory reactions via inhibiting pro-inflammatory mediator release and/or by acting at post-junctional targets on the vascular endothelium.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acute Disease
  • Animals
  • Capsaicin / administration & dosage
  • Capsaicin / toxicity
  • Carrageenan / administration & dosage
  • Carrageenan / toxicity
  • Diterpenes / administration & dosage
  • Diterpenes / toxicity
  • Edema / chemically induced
  • Edema / prevention & control
  • Inflammation / blood*
  • Inflammation / chemically induced
  • Injections, Intraperitoneal
  • Male
  • Mass Spectrometry
  • Neurogenic Inflammation / blood*
  • Neurogenic Inflammation / chemically induced
  • Pituitary Adenylate Cyclase-Activating Polypeptide / administration & dosage
  • Pituitary Adenylate Cyclase-Activating Polypeptide / blood*
  • Pituitary Adenylate Cyclase-Activating Polypeptide / pharmacology
  • Radioimmunoassay
  • Rats
  • Rats, Wistar
  • TRPV Cation Channels / antagonists & inhibitors

Substances

  • Diterpenes
  • Pituitary Adenylate Cyclase-Activating Polypeptide
  • TRPV Cation Channels
  • Trpv1 protein, rat
  • Carrageenan
  • resiniferatoxin
  • Capsaicin