Wnt4 inhibits beta-catenin/TCF signalling by redirecting beta-catenin to the cell membrane

Biol Cell. 2008 Mar;100(3):167-77. doi: 10.1042/BC20070072.

Abstract

Background information: During embryonic development, beta-catenin is central both to the transcriptional activation of Wnt [wingless-type MMTV (murine-mammary-tumour virus) integration site family] target genes and as a mediator of cell-cell adhesion. Signals that regulate its levels and subcellular localization are critical. One mechanism of Wnt signalling results in stabilization of beta-catenin protein, which leads to its translocation into the nucleus, where it interacts with TCF (T-cell factor, HMG box) and activates transcription of target genes. Less well understood are mechanisms of Wnt signalling that do not involve beta-catenin stabilization and result in inhibition of beta-catenin-mediated transcription.

Results: Here, we show that a member of the Wnt protein family, Wnt4 (Wnt, member 4), regulates the subcellular localization of beta-catenin, redirecting it to the cell membrane. Unique among Wnts, this action does not affect the stability of beta-catenin but does prohibit its involvement in TCF gene transactivation.

Conclusions: This novel mechanism suggests that Wnt4 acts as a switch between the two modes of beta-catenin function, transcriptional activation and cell-cell adhesion.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cell Adhesion / genetics
  • Cell Communication / genetics
  • Cell Line
  • Cell Membrane / genetics
  • Cell Membrane / metabolism*
  • Gene Expression Regulation / genetics
  • Humans
  • Mice
  • Mice, Knockout
  • Protein Transport / physiology
  • Signal Transduction / genetics*
  • TCF Transcription Factors / genetics
  • TCF Transcription Factors / metabolism*
  • Transcriptional Activation / genetics
  • Wnt Proteins / genetics
  • Wnt Proteins / metabolism*
  • Wnt4 Protein
  • beta Catenin / genetics
  • beta Catenin / metabolism*

Substances

  • CTNNB1 protein, mouse
  • TCF Transcription Factors
  • WNT4 protein, human
  • Wnt Proteins
  • Wnt4 Protein
  • Wnt4 protein, mouse
  • beta Catenin