Decoralin, a novel linear cationic alpha-helical peptide from the venom of the solitary eumenine wasp Oreumenes decoratus

Peptides. 2007 Dec;28(12):2320-7. doi: 10.1016/j.peptides.2007.09.017. Epub 2007 Sep 29.

Abstract

A novel peptide, decoralin, was isolated from the venom of the solitary eumenine wasp Oreumenes decoratus. Its sequence, Ser-Leu-Leu-Ser-Leu-Ile-Arg-Lys-Leu-Ile-Thr, was determined by Edman degradation and corroborated by solid-phase synthesis. This sequence has the characteristic features of linear cationic alpha-helical peptides; rich in hydrophobic and basic amino acids with no disulfide bond, and accordingly, it can be predicted to adopt an amphipathic alpha-helix secondary structure. In fact, the CD spectra of decoralin in the presence of TFE or SDS showed a high alpha-helical conformation content. In a biological evaluation, decoralin exhibited a significant broad-spectrum antimicrobial activity, and moderate mast cell degranulation and leishmanicidal activities, but showed virtually no hemolytic activity. A synthetic analog with C-terminal amidation showed a much more potent activity in all the biological assays.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Antimicrobial Cationic Peptides / chemistry
  • Antimicrobial Cationic Peptides / genetics
  • Antimicrobial Cationic Peptides / isolation & purification
  • Antimicrobial Cationic Peptides / pharmacology
  • Bacteria / drug effects
  • Cell Degranulation / drug effects
  • Circular Dichroism
  • Hemolysis / drug effects
  • Humans
  • In Vitro Techniques
  • Mast Cells / drug effects
  • Mast Cells / physiology
  • Mice
  • Oligopeptides / chemistry*
  • Oligopeptides / genetics
  • Oligopeptides / isolation & purification*
  • Oligopeptides / pharmacology
  • Protein Structure, Secondary
  • Rats
  • Wasp Venoms / chemistry*
  • Wasp Venoms / genetics
  • Wasp Venoms / pharmacology
  • Wasps / chemistry
  • Wasps / genetics

Substances

  • Antimicrobial Cationic Peptides
  • Oligopeptides
  • Wasp Venoms