A hypoallergenic vaccine obtained by tail-to-head restructuring of timothy grass pollen profilin, Phl p 12, for the treatment of cross-sensitization to profilin

J Immunol. 2007 Dec 1;179(11):7624-34. doi: 10.4049/jimmunol.179.11.7624.

Abstract

Profilins are highly cross-reactive allergens in pollens and plant food. In a paradigmatic approach, the cDNA coding for timothy grass pollen profilin, Phl p 12, was used as a template to develop a new strategy for engineering an allergy vaccine with low IgE reactivity. Non-IgE-reactive fragments of Phl p 12 were identified by synthetic peptide chemistry and restructured (rs) as a new molecule, Phl p 12-rs. It comprised the C terminus of Phl p 12 at its N terminus and the Phl p 12 N terminus at its C terminus. Phl p 12-rs was expressed in Escherichia coli and purified to homogeneity. Determination of secondary structure by circular dichroism indicated that the restructuring process had reduced the IgE-reactive alpha-helical contents of the protein but retained its beta-sheet conformation. Phl p 12-rs exhibited reduced IgE binding capacity and allergenic activity but preserved T cell reactivity in allergic patients. IgG Abs induced by immunization of mice and rabbits with Phl p 12-rs cross-reacted with pollen and food-derived profilins. Recombinant Phl p 12-rs, rPhl p 12-rs, induced less reaginic IgE to the wild-type allergen than rPhl p 12. However, the rPhl p 12-rs-induced IgGs inhibited allergic patients' IgE Ab binding to profilins to a similar degree as those induced by immunization with the wild type. Phl p 12-rs specific IgG inhibited profilin-induced basophil degranulation. In conclusion, a restructured recombinant vaccine was developed for the treatment of profilin-allergic patients. The strategy of tail-to-head reassembly of hypoallergenic allergen fragments within one molecule represents a generally applicable strategy for the generation of allergy vaccines.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Allergens / chemistry
  • Allergens / genetics
  • Allergens / immunology*
  • Anti-Allergic Agents / chemistry
  • Anti-Allergic Agents / immunology*
  • Antibodies / chemistry
  • Antibodies / genetics
  • Antibodies / immunology
  • Antibody Specificity / genetics
  • Antibody Specificity / immunology
  • Antigen-Antibody Reactions
  • Antigens, Plant / chemistry
  • Antigens, Plant / genetics
  • Antigens, Plant / immunology*
  • Binding Sites
  • Circular Dichroism
  • Epitopes / immunology
  • Genetic Engineering / methods
  • Histamine / immunology
  • Humans
  • Immunoglobulin E / blood
  • Immunoglobulin E / immunology
  • Immunoglobulin G / blood
  • Immunoglobulin G / immunology
  • Models, Molecular
  • Pollen / chemistry
  • Pollen / genetics
  • Pollen / immunology*
  • Polymerase Chain Reaction
  • Profilins / chemistry
  • Profilins / genetics
  • Profilins / immunology*
  • Protein Structure, Secondary
  • Recombinant Fusion Proteins / chemistry
  • Recombinant Fusion Proteins / genetics
  • Recombinant Fusion Proteins / immunology*
  • Sensitivity and Specificity
  • T-Lymphocytes / immunology
  • Vaccines / chemistry
  • Vaccines / genetics
  • Vaccines / immunology*

Substances

  • Allergens
  • Anti-Allergic Agents
  • Antibodies
  • Antigens, Plant
  • Epitopes
  • Immunoglobulin G
  • Phl p 12 allergen, timothy grass
  • Profilins
  • Recombinant Fusion Proteins
  • Vaccines
  • Immunoglobulin E
  • Histamine