Activation of p53-dependent responses in tumor cells treated with a PARC-interacting peptide

Biochem Biophys Res Commun. 2008 Apr 4;368(2):350-6. doi: 10.1016/j.bbrc.2008.01.093. Epub 2008 Jan 28.

Abstract

We tested the activity of a p53 carboxy-terminal peptide containing the PARC-interacting region in cancer cells with wild type cytoplasmic p53. Peptide delivery was achieved by fusing it to the TAT transduction domain (TAT-p53-C-ter peptide). In a two-hybrid assay, the tetramerization domain (TD) of p53 was necessary and sufficient to bind PARC. The TAT-p53-C-ter peptide disrupted the PARC-p53 complex. Peptide treatment caused p53 nuclear relocation, p53-dependent changes in gene expression and enhancement of etoposide-induced apoptosis. These studies suggest that PARC-interacting peptides are promising candidates for the enhancement of p53-dependent apoptosis in tumors with wt cytoplasmic p53.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Apoptosis / drug effects*
  • Cell Line, Tumor
  • DNA Topoisomerase IV / administration & dosage*
  • Humans
  • Neoplasms / metabolism*
  • Neoplasms / pathology*
  • Signal Transduction / drug effects*
  • Tumor Suppressor Protein p53 / metabolism*

Substances

  • TP53 protein, human
  • Tumor Suppressor Protein p53
  • DNA Topoisomerase IV