Calcium regulation of myogenesis by differential calmodulin inhibition of basic helix-loop-helix transcription factors

Mol Biol Cell. 2008 Jun;19(6):2509-19. doi: 10.1091/mbc.e07-09-0886. Epub 2008 Mar 19.

Abstract

The members of the MyoD family of basic helix-loop-helix (bHLH) transcription factors are critical regulators of skeletal muscle differentiation that function as heterodimers with ubiquitously expressed E-protein bHLH transcription factors. These heterodimers must compete successfully with homodimers of E12 and other E-proteins to enable myogenesis. Here, we show that E12 mutants resistant to Ca(2+)-loaded calmodulin (CaM) inhibit MyoD-initiated myogenic conversion of transfected fibroblasts. Ca(2+) channel blockers reduce, and Ca(2+) stimulation increases, transcription by coexpressed MyoD and wild-type E12 but not CaM-resistant mutant E12. Furthermore, CaM-resistant E12 gives lower MyoD binding and higher E12 binding to a MyoD-responsive promoter in vivo and cannot rescue myogenic differentiation that has been inhibited by siRNA against E12 and E47. Our data support the concept that Ca(2+)-loaded CaM enables myogenesis by inhibiting DNA binding of E-protein homodimers, thereby promoting occupancy of myogenic bHLH protein/E-protein heterodimers on promoters of myogenic target genes.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Animals
  • Basic Helix-Loop-Helix Transcription Factors / antagonists & inhibitors*
  • Basic Helix-Loop-Helix Transcription Factors / chemistry
  • Calcium / metabolism*
  • Calmodulin / metabolism*
  • Cell Differentiation
  • Cell Nucleus / metabolism
  • Dimerization
  • Genes, Reporter
  • Mice
  • Molecular Sequence Data
  • Muscle Development*
  • Mutant Proteins / metabolism
  • Mutation / genetics
  • MyoD Protein / genetics
  • MyoD Protein / metabolism
  • NIH 3T3 Cells
  • Promoter Regions, Genetic / genetics
  • RNA, Small Interfering / metabolism
  • Rats
  • Recombinant Fusion Proteins / metabolism
  • TCF Transcription Factors / antagonists & inhibitors*
  • TCF Transcription Factors / chemistry
  • Transcription Factor 7-Like 1 Protein
  • Transcriptional Activation
  • Transfection

Substances

  • Basic Helix-Loop-Helix Transcription Factors
  • Calmodulin
  • Mutant Proteins
  • MyoD Protein
  • RNA, Small Interfering
  • Recombinant Fusion Proteins
  • TCF Transcription Factors
  • Tcf7l1 protein, mouse
  • Transcription Factor 7-Like 1 Protein
  • Calcium