High doses of lercanidipine are better tolerated than other dihydropyridines in hypertensive patients with metabolic syndrome: results from the TOLERANCE study

Int J Clin Pract. 2008 May;62(5):723-8. doi: 10.1111/j.1742-1241.2008.01736.x. Epub 2008 Mar 17.

Abstract

Aims/introduction: The TOlerabilidad de LERcanidipino 20 mg frente a Amlodipino y Nifedipino en CondicionEs normales de uso study was aimed to compare the tolerability of high doses of lercanidipine with amlodipine and nifedipine gastro-intestinal therapeutic system (GITS) in the treatment of hypertension in daily clinical practice.

Patients/methods: Essential hypertensives >or= 18 years, treated during at least 1 month with lercanidipine 20 mg, amlodipine 10 mg or nifedipine GITS 60 mg, after a previous treatment course of at least 1 month with half the dose of the corresponding drugs were included. We present the data of the subgroup of patients with metabolic syndrome (MetS).

Results: Three hundred and thirty-seven of the 650 study population fulfilled criteria of MetS, 233 (69.1%) on lercanidipine and 104 (30.9%) on amlodipine/nifedipine GITS. Overall, a significantly lower proportion of lercanidipine-treated patients showed adverse reactions (ARs) when compared with patients receiving other-dihydropyridines (DHPs) (60.1% vs. 73.1%, p = 0.003). Similarly, the most common vasodilation-related ARs (oedema, swelling, flushing and headache) were significantly less frequent in lercanidipine group (all p < 0.01).

Conclusion: In conclusion, lercanidipine appears to exhibit a better tolerability profile and less vasodilation-related ARs compared with other DHPs in hypertensive patients with MetS.

Publication types

  • Clinical Trial
  • Multicenter Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adolescent
  • Adult
  • Aged
  • Amlodipine / adverse effects
  • Amlodipine / therapeutic use
  • Antihypertensive Agents / administration & dosage*
  • Antihypertensive Agents / adverse effects
  • Calcium Channel Blockers / adverse effects
  • Calcium Channel Blockers / therapeutic use
  • Cross-Sectional Studies
  • Dihydropyridines / administration & dosage*
  • Dihydropyridines / adverse effects
  • Dose-Response Relationship, Drug
  • Female
  • Humans
  • Hypertension / drug therapy*
  • Male
  • Metabolic Syndrome / drug therapy*
  • Middle Aged
  • Nifedipine / adverse effects
  • Nifedipine / therapeutic use

Substances

  • Antihypertensive Agents
  • Calcium Channel Blockers
  • Dihydropyridines
  • Amlodipine
  • Nifedipine
  • lercanidipine