The essential role of fibroblasts in esophageal squamous cell carcinoma-induced angiogenesis

Gastroenterology. 2008 Jun;134(7):1981-93. doi: 10.1053/j.gastro.2008.02.061. Epub 2008 Mar 4.

Abstract

Background & aims: Esophageal squamous cell carcinoma (ESCC) is known to be a highly angiogenic tumor. Here, we investigated the role of the stromal fibroblasts in the ESCC-induced angiogenic response using a novel 3-dimensional model.

Methods: A novel assay was developed where cocultures of ESCC and esophageal fibroblasts induced human microvascular endothelial cell (HMVEC) vascular network formation in a 3-dimensional collagen gel. Biochemical studies showed that the ESCC-induced activation of the fibroblasts was required to induce vascular network formation via a transforming growth factor (TGF)-beta and vascular endothelial growth factor (VEGF)-dependent pathway.

Results: Conditioned media from a panel of 4 ESCC lines transdifferentiated normal esophageal fibroblasts into myofibroblasts via TGF-beta signaling. The presence of fibroblasts was essential for efficient HMVEC network formation, and the addition of ESCC cells to these cultures greatly enhanced the angiogenic process. The role of TGF-beta in this process was shown by the complete inhibition of network formation following TGF-beta inhibitor treatment. Finally, we showed that ESCC-derived TGF-beta regulates angiogenesis through the release of VEGF from the fibroblasts and that the VEGF release was blocked following TGF-beta inhibition.

Conclusions: This study shows the essential role of fibroblasts in the ESCC angiogenic-induced response and suggests that the pharmacologic targeting of the TGF-beta signaling axis could be of therapeutic benefit in this deadly disease.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Benzamides / pharmacology
  • Benzodioxoles / pharmacology
  • Carcinoma, Squamous Cell / blood supply
  • Carcinoma, Squamous Cell / metabolism*
  • Cell Line, Tumor
  • Cell Transdifferentiation
  • Coculture Techniques
  • Collagen / metabolism
  • Culture Media, Conditioned / metabolism
  • Dose-Response Relationship, Drug
  • Endothelial Cells / drug effects
  • Endothelial Cells / metabolism*
  • Esophageal Neoplasms / blood supply
  • Esophageal Neoplasms / metabolism*
  • Esophagus / embryology
  • Esophagus / metabolism
  • Fibroblasts / drug effects
  • Fibroblasts / metabolism*
  • Fibroblasts / pathology
  • Gels
  • Humans
  • Imidazoles / pharmacology
  • Microcirculation / metabolism
  • Neovascularization, Pathologic / metabolism*
  • Paracrine Communication* / drug effects
  • Pyrazoles / pharmacology
  • Pyridines / pharmacology
  • Transfection
  • Transforming Growth Factor beta1 / antagonists & inhibitors
  • Transforming Growth Factor beta1 / metabolism
  • Transforming Growth Factor beta2 / metabolism
  • Vascular Endothelial Growth Factor A / metabolism

Substances

  • 2-(5-benzo(1,3)dioxol-5-yl-2-tert-butyl-3H-imidazol-4-yl)-6-methylpyridine hydrochloride
  • 4-(4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)pyridin-2-yl)-N-(tetrahydro-2H-pyran-4-yl)benzamide
  • Benzamides
  • Benzodioxoles
  • Culture Media, Conditioned
  • Gels
  • Imidazoles
  • Pyrazoles
  • Pyridines
  • Transforming Growth Factor beta1
  • Transforming Growth Factor beta2
  • VEGFA protein, human
  • Vascular Endothelial Growth Factor A
  • Collagen