Analysis of Ret knockin mice reveals a critical role for IKKs, but not PI 3-K, in neurotrophic factor-induced survival of sympathetic neurons

Cell Death Differ. 2008 Sep;15(9):1510-21. doi: 10.1038/cdd.2008.76. Epub 2008 May 23.

Abstract

We analyzed the survival responses and downstream signaling elicited by GDNF on sympathetic neurons from different Ret knockin mice. Lack of tyrosine 1062, a multidocking site in Ret, completely prevented GDNF-mediated survival. Importantly, lack of tyrosine 981, although abrogating Akt phosphorylation, had no effect on neuronal survival, indicating that the PI 3-K/Akt pathway is not necessary for survival of sympathetic neurons. In contrast, silencing of B-Raf completely prevented not only GDNF-mediated but also NGF-mediated cell survival, independently of MEK-1/2. We identified IKKs as the main effectors of the protective effects of B-Raf. First, B-Raf interacted with and activated IKKs. Second, knockdown of IKKs reversed the protection afforded by a constitutively active form of B-Raf. Third, knockdown of IKKs prevented both NGF- and GDNF-mediated survival. In conclusion, our data delineate a novel survival pathway for sympathetic neurons linking B-Raf to IKKs, independently of both PI 3-K and MEK-1/2 pathways.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cell Size
  • Cell Survival
  • Cells, Cultured
  • Extracellular Signal-Regulated MAP Kinases / metabolism
  • Glial Cell Line-Derived Neurotrophic Factor / pharmacology*
  • Humans
  • I-kappa B Kinase / physiology*
  • Mice
  • Mice, Mutant Strains
  • Mutation
  • Nerve Growth Factor / pharmacology
  • Neurons / cytology
  • Neurons / drug effects
  • Neurons / enzymology*
  • Phosphatidylinositol 3-Kinases / physiology*
  • Proto-Oncogene Proteins B-raf / metabolism
  • Proto-Oncogene Proteins c-akt / metabolism
  • Proto-Oncogene Proteins c-ret / chemistry
  • Proto-Oncogene Proteins c-ret / genetics
  • Proto-Oncogene Proteins c-ret / metabolism*
  • Signal Transduction
  • Sympathetic Nervous System / cytology
  • Tyrosine / genetics

Substances

  • Glial Cell Line-Derived Neurotrophic Factor
  • Tyrosine
  • Nerve Growth Factor
  • Phosphatidylinositol 3-Kinases
  • Proto-Oncogene Proteins c-ret
  • RET protein, human
  • Proto-Oncogene Proteins B-raf
  • Proto-Oncogene Proteins c-akt
  • I-kappa B Kinase
  • Extracellular Signal-Regulated MAP Kinases