RhoA-GDP regulates RhoB protein stability. Potential involvement of RhoGDIalpha

J Biol Chem. 2008 Aug 1;283(31):21588-98. doi: 10.1074/jbc.M710033200. Epub 2008 Jun 4.

Abstract

RhoA plays a significant role in actin stress fibers formation. However, silencing RhoA alone or RhoA and RhoC did not completely suppress the stress fibers suggesting a residual "Rho-like" activity. RhoB, the third member of the Rho subclass, is a shortlived protein barely detectable in basal conditions. In various cell types, the silencing of RhoA induced a strong up-regulation of both total and active RhoB protein levels that were rescued by re-expressing RhoA and related to an enhanced half-life of the protein. The RhoA-dependent regulation of RhoB does not depend on the activity of RhoA but is mediated by its GDP-bound form. The stabilization of RhoB was not dependent on isoprenoid biosynthesis, Rho kinase, extracellular signal-regulated kinase, p38 mitogen-activated kinase, or phosphatidylinositol 3'-OH kinase pathways but required RhoGDIalpha. The forced expression of RhoGDIalpha increased RhoB half-life, whereas its knock-down antagonized the induction of RhoB following RhoA silencing. Moreover, a RhoA mutant (RhoAR68E) unable to bind RhoGDIalpha was significantly less efficient as compared with wild-type RhoA in reversing RhoB up-regulation upon RhoA silencing. These results suggest that, in basal conditions, RhoGDIalpha is rate-limiting and the suppression of RhoA makes it available to stabilize RhoB. Our results highlight RhoGDIalpha-dependent cross-talks that regulate the stability of RhoGTPases.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Gene Silencing
  • Genetic Vectors
  • Guanine Nucleotide Dissociation Inhibitors / metabolism*
  • Guanosine Diphosphate / chemistry*
  • Humans
  • Models, Biological
  • Protein Transport
  • Reverse Transcriptase Polymerase Chain Reaction
  • Signal Transduction
  • Transfection
  • Up-Regulation
  • rho GTP-Binding Proteins / metabolism
  • rho-Specific Guanine Nucleotide Dissociation Inhibitors
  • rhoA GTP-Binding Protein / metabolism
  • rhoA GTP-Binding Protein / physiology*
  • rhoB GTP-Binding Protein / metabolism*
  • rhoC GTP-Binding Protein

Substances

  • Guanine Nucleotide Dissociation Inhibitors
  • rho-Specific Guanine Nucleotide Dissociation Inhibitors
  • Guanosine Diphosphate
  • RHOC protein, human
  • rho GTP-Binding Proteins
  • rhoA GTP-Binding Protein
  • rhoB GTP-Binding Protein
  • rhoC GTP-Binding Protein