Pharmacotherapy of essential thrombocythemia

Expert Opin Pharmacother. 2008 Jul;9(10):1679-85. doi: 10.1517/14656566.9.10.1679.

Abstract

Background: The natural history of essential thrombocythemia is characterized by an increased incidence of thrombotic and hemorrhagic events and, in the long-term, a tendency for disease transformation to myelofibrosis or acute leukemia. Advanced age and a prior history of thrombosis are the major predictors of thrombotic complications.

Objective: The aim of this study was to outline the current evidence and the authors' opinion regarding the clinical management of patients with essential thrombocythemia.

Methods: The study reviewed the pertinent literature addressing the management options for essential thrombocythemia patients.

Results/conclusions: Cytoreductive agents can reduce the rate of thrombotic events, but do not affect the overall survival or rate of disease transformation. Thus, a risk-adapted strategy is recommended for the management of patients with essential thrombocythemia. High-risk patients with essential thrombocythemia should be treated with cytoreductive therapy and low-dose aspirin. Hydroxycarbamide is the agent of choice in most patients: however, interferon-alpha is a reasonable alternative in young patients, pregnancy or those intolerant of hydroxycarbamide. Low-risk patients can be safely observed. The management of intermediate-risk patients needs to be individualized: however, low-dose aspirin can be used after excluding acquired von Willebrand's disease. In the future we await the role of molecularly targeted therapy with JAK2 inhibitors in high-risk essential thrombocythemia patients.

Publication types

  • Review

MeSH terms

  • Age Factors
  • Antineoplastic Agents / therapeutic use
  • Aspirin / therapeutic use
  • Disease Progression
  • Humans
  • Hydroxyurea / therapeutic use
  • Interferon-alpha / therapeutic use
  • Janus Kinase 2 / antagonists & inhibitors
  • Platelet Aggregation Inhibitors / therapeutic use*
  • Risk Factors
  • Thrombocythemia, Essential / blood
  • Thrombocythemia, Essential / drug therapy*

Substances

  • Antineoplastic Agents
  • Interferon-alpha
  • Platelet Aggregation Inhibitors
  • Janus Kinase 2
  • Aspirin
  • Hydroxyurea