Lethal damage to murine L1210 cells by exogenous lipid hydroperoxides: protective role of glutathione-dependent selenoperoxidases

Arch Biochem Biophys. 1991 Aug 1;288(2):671-80. doi: 10.1016/0003-9861(91)90250-m.

Abstract

The effect of selenium deprivation on the viability of murine L1210 cells exposed to various exogenous lipid hydroperoxides has been investigated. Selenoperoxidase activities of cells grown for longer than 1 week in 1% serum with no added selenium [Se(-) cells] were less than 10% of the activities of selenium-satisfied controls [Se(+) cells] or selenium-repleted counterparts [Se(-/+) cells]. The enzymes measured were classical glutathione peroxidase (GPX) and phospholipid hydroperoxide glutathione peroxidase (PHGPX). Se(-) cells exhibited a compensatory increase in catalase activity. Dye exclusion and clonal survival assays indicated that Se(-) and Se(+) cells were relatively insensitive to photochemically generated phospholipid hydroperoxides in liposomal form. However, both cell types were sensitive to liposomal cholesterol hydroperoxides, e.g., 7-hydroperoxycholesterol (7-OOH), Se(-) being much more so (LD50 approximately 10 microM) than Se(+) (LD50 approximately 75 microM). By contrast, 7-hydroxycholesterol over a comparable concentration range was minimally toxic to Se(-) and Se(+) cells. Cell killing by 7-OOH was inhibited by desferrioxamine and by butylated hydroxytoluene, suggesting that iron-mediated free radical reactions are involved. The involvement of glutathione in cytoprotection was confirmed by showing that Se(+) cells were more sensitive to 7-OOH after treating with buthionine sulfoximine, an inhibitor of GSH synthesis. Cellular detoxification of 7-OOH is provisionally attributed to PHGPX rather than GPX, since 7-OOH and other cholesterol hydroperoxides were found to be good substrates for PHGPX in a cell free system, but were unreactive with GPX.

Publication types

  • Comparative Study
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Animals
  • Butylated Hydroxytoluene / pharmacology
  • Cell Survival / drug effects*
  • Cell-Free System
  • Cholesterol / analogs & derivatives*
  • Cholesterol / metabolism
  • Cholesterol / pharmacology
  • Deferoxamine / pharmacology
  • Dose-Response Relationship, Drug
  • Glutathione Peroxidase / metabolism*
  • Kinetics
  • Leukemia L1210 / enzymology
  • Leukemia L1210 / pathology*
  • Lipid Peroxides / pharmacology*
  • Liposomes
  • Mice
  • Phospholipids / metabolism
  • Selenium / pharmacology*

Substances

  • Lipid Peroxides
  • Liposomes
  • Phospholipids
  • Butylated Hydroxytoluene
  • cholesterol 7-hydroperoxide
  • Cholesterol
  • Glutathione Peroxidase
  • Selenium
  • Deferoxamine