(-)-Epigallocatechin-3-gallate prevents lipopolysaccharide-induced elevation of beta-amyloid generation and memory deficiency

Brain Res. 2009 Jan 23:1250:164-74. doi: 10.1016/j.brainres.2008.10.012. Epub 2008 Nov 1.

Abstract

Neuroinflammation has been known to play a role in the pathogenesis of AD. Our previous study showed that lipopolysaccharide (LPS) induced memory impairment through the accumulation of Abeta via the increase of beta- and gamma-secretase. In this study, we investigated the possible preventive effect of (-)-epigallocatechin-3-gallate (EGCG) on memory deficiency caused by LPS through the inhibition of Abeta(1-42) generation. Oral treatment with EGCG (1.5 and 3 mg/kg, for 3 weeks) into drinking water ameliorated LPS (1 microg/mouse, i.c.v.)-induced memory deficiency in a dose dependent manner. In addition, EGCG also dose-dependently inhibited LPS-induced elevation of Abeta level through attenuation of LPS-induced beta- and gamma-secretase activities and expression of its metabolic products; C99 and Abeta. Moreover, EGCG prevented LPS-induced neuronal cell death as well as the expression of inflammatory proteins, inducible nitric oxide synthetase and cyclooxygenase-2. This study therefore suggests that EGCG prevents LPS-mediated apoptotic cell death through the inhibition of the elevation of Abeta via the inhibition of beta- and gamma-secretases, and thus EGCG can be a useful agent against neuroinflammation-associated development or progression of AD.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amyloid Precursor Protein Secretases / metabolism
  • Amyloid beta-Peptides / metabolism*
  • Animals
  • Apoptosis / drug effects
  • Avoidance Learning / drug effects
  • Brain / drug effects
  • Brain / metabolism*
  • Catechin / administration & dosage
  • Catechin / analogs & derivatives*
  • Catechin / pharmacology
  • Cerebral Cortex / drug effects
  • Cerebral Cortex / metabolism
  • Cyclooxygenase 2 / metabolism
  • Glial Fibrillary Acidic Protein
  • Hippocampus / drug effects
  • Hippocampus / metabolism
  • Lipopolysaccharides*
  • Male
  • Maze Learning / drug effects
  • Memory / drug effects*
  • Memory Disorders / physiopathology
  • Memory Disorders / prevention & control*
  • Mice
  • Nerve Tissue Proteins / metabolism
  • Neurons / drug effects
  • Neurons / metabolism
  • Nitric Oxide Synthase Type II / metabolism
  • Peptide Fragments / metabolism

Substances

  • Amyloid beta-Peptides
  • Glial Fibrillary Acidic Protein
  • Lipopolysaccharides
  • Nerve Tissue Proteins
  • Peptide Fragments
  • amyloid beta-protein (1-42)
  • glial fibrillary astrocytic protein, mouse
  • Catechin
  • epigallocatechin gallate
  • Nitric Oxide Synthase Type II
  • Ptgs2 protein, mouse
  • Cyclooxygenase 2
  • Amyloid Precursor Protein Secretases