Switch-like control of SREBP-2 transport triggered by small changes in ER cholesterol: a delicate balance

Cell Metab. 2008 Dec;8(6):512-21. doi: 10.1016/j.cmet.2008.10.008.

Abstract

Animal cells control their membrane lipid composition within narrow limits, but the sensing mechanisms underlying this control are largely unknown. Recent studies disclosed a protein network that controls the level of one lipid-cholesterol. This network resides in the endoplasmic reticulum (ER). A key component is Scap, a tetrameric ER membrane protein that binds cholesterol. Cholesterol binding prevents Scap from transporting SREBPs to the Golgi for activation. Using a new method to purify ER membranes from cultured cells, we show that Scap responds cooperatively to ER cholesterol levels. When ER cholesterol exceeds 5% of total ER lipids (molar basis), SREBP-2 transport is abruptly blocked. Transport resumes when ER cholesterol falls below the 5% threshold. The 5% threshold is lowered to 3% when cells overexpress Insig-1, a Scap-binding protein. Cooperative interactions between cholesterol, Scap, and Insig create a sensitive switch that controls the cholesterol composition of cell membranes with remarkable precision.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Biological Transport
  • CHO Cells
  • Cells, Cultured
  • Cholesterol / metabolism*
  • Cricetinae
  • Cricetulus
  • Endoplasmic Reticulum / metabolism*
  • Golgi Apparatus / metabolism
  • Mass Spectrometry
  • Protein Processing, Post-Translational
  • Sterol Regulatory Element Binding Protein 2 / biosynthesis
  • Sterol Regulatory Element Binding Protein 2 / metabolism*
  • Time Factors

Substances

  • SREBF2 protein, human
  • Sterol Regulatory Element Binding Protein 2
  • Cholesterol