Edaravone, a novel free radical scavenger, reduces high-mobility group box 1 and prolongs survival in a neonatal sepsis model

Shock. 2009 Dec;32(6):586-92. doi: 10.1097/SHK.0b013e3181a2b886.

Abstract

Free radicals play an important role in the inflammatory process of sepsis. We hypothesized that edaravone, a novel free radical scavenger, can suppress pathophysiological events and prolong survival in a neonatal sepsis cecal ligation and perforation (CLP) model. Of 32 3-day-old anesthetized and mechanically ventilated piglets, 11 received CLP only, 10 received CLP and edaravone treatment starting 30 min after CLP, and 11 constituted a sham (control) group. Mean arterial pressure (MAP), heart rate, cardiac output, arterial blood gas, serum total hydroperoxide, nitrite and nitrate, TNF-alpha, and high-mobility group box 1 (HMGB1) were measured before CLP and at 1, 3, and 6 h after CLP. Compared with the CLP group, the edaravone group showed higher MAP at 6 h, lower heart rate at 1 and 3 h, lower total hydroperoxide at 1 h, lower nitrite and nitrate at 3 and 6 h, and higher (although not significantly so) mean cardiac output at 1, 3, and 6 h. TNF-alpha elevation was delayed from 1 h in the CLP group to 3 h in the edaravone group. In the edaravone group, HMGB1 did not change significantly at any time, whereas in the CLP group, it increased at 6 h. Survival times were longer in the edaravone group than in the CLP group (15.4 +/- 1.4 vs. 10.2 +/- 1 h; P < 0.005). In addition, each of the serial dilutions of edaravone had a higher biological antioxidant potential than tempol does. In conclusion, edaravone suppressed free radicals, delayed the TNF-alpha surge, and prevented HMGB1 elevation, thereby maintaining MAP and prolonging survival time in a neonatal sepsis CLP model.

MeSH terms

  • Animals
  • Animals, Newborn
  • Antioxidants / chemistry
  • Antipyrine / analogs & derivatives*
  • Antipyrine / pharmacology
  • Blood Pressure
  • Body Weight
  • Cyclic N-Oxides / pharmacology
  • Edaravone
  • Free Radical Scavengers / pharmacology*
  • Free Radicals
  • HMGB1 Protein / blood*
  • Heart Rate
  • Inflammation
  • Sepsis / physiopathology*
  • Spin Labels
  • Swine
  • Time Factors

Substances

  • Antioxidants
  • Cyclic N-Oxides
  • Free Radical Scavengers
  • Free Radicals
  • HMGB1 Protein
  • Spin Labels
  • Edaravone
  • Antipyrine
  • tempol