Liver X receptors interfere with cytokine-induced proliferation and cell survival in normal and leukemic lymphocytes

J Leukoc Biol. 2009 Nov;86(5):1039-48. doi: 10.1189/jlb.1008663. Epub 2009 Aug 11.

Abstract

Liver X receptors (LXRs) are nuclear receptors regulating lipid and cholesterol metabolism. Recent data indicate an additional role of LXR in immunity by controlling dendritic cell and T-cell function and in breast and prostate cancer cells. Here, we show that LXR activation interferes with IL-2 and IL-7-induced proliferation and cell cycle progression of human T-cell blasts mainly through inhibited phosphorylation of the retinoblastoma protein and decreased expression of the cell cycle protein cyclin B. Comparable results were obtained with IL-2-dependent chronic lymphoblastic leukemia (CLL) T cells. Furthermore, we show for B-CLL cells that LXR are functionally active and inhibit expression of survival genes bcl-2 and MMP-9, and significantly reduce cell viability, suggesting an interference of LXR with cytokine-dependent CLL cell survival. In conclusion, our data reveal LXR as a potent modulator of cytokine-dependent proliferation and survival of normal and malignant T and B lymphocytes. This novel LXR action could find clinical application in immunosuppressive and antileukemic therapies.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antigens, CD / immunology
  • Cell Division / drug effects
  • Cell Survival / drug effects
  • Cholesterol / metabolism
  • Cytokines / pharmacology*
  • Humans
  • Leukemia / immunology
  • Leukemia / pathology*
  • Leukemia, Lymphocytic, Chronic, B-Cell / immunology*
  • Leukemia, Lymphocytic, Chronic, B-Cell / pathology
  • Leukemia, Prolymphocytic, T-Cell / immunology
  • Leukemia, Prolymphocytic, T-Cell / pathology
  • Lipids / physiology
  • Liver X Receptors
  • Lymphocytes / cytology
  • Lymphocytes / drug effects
  • Lymphocytes / immunology*
  • Lymphocytes / pathology*
  • Methylphenazonium Methosulfate / pharmacology
  • Orphan Nuclear Receptors / immunology
  • Orphan Nuclear Receptors / physiology*
  • T-Lymphocytes / immunology

Substances

  • Antigens, CD
  • Cytokines
  • Lipids
  • Liver X Receptors
  • Orphan Nuclear Receptors
  • Methylphenazonium Methosulfate
  • Cholesterol