Effects of monthly intramuscular neridronate in rheumatic patients in chronic treatment with low-dose glucocorticoids

Clin Exp Rheumatol. 2009 Jul-Aug;27(4):567-73.

Abstract

Objectives: To assess the effects of intramuscular (im) neridronate (NE) on lumbar and femoral neck BMD and on markers of bone turnover in rheumatic patients under chronic low-dose glucocorticoids (GC) therapy.

Methods: Sixty-nine osteopoenic and osteoporotic patients, affected by rheumatic diseases and gastric or esophageal conditions which contraindicated treatment with oral bisphosphonates (BPs), were randomly assigned to: Group A (23 patients) administered with daily calcium 1 g and vitamin D 800 UI; Group B (46 patients) receiving daily calcium 1 g, vitamin D 800 UI and im NE 25 mg monthly.

Results: After 12 months of therapy (M12) lumbar BMD was reduced of 2.97% in Group A, and improved of 3.34% (p=0.001) in Group B; at M12, femoral neck BMD was reduced of 2.40% in Group A and improved of 1.78% in Group B (p=0.010). After 6 (M6) and 12 months of therapy, the bone resorption markers were significantly reduced in Group B: OHPr-41.64% at M6 (p<0.001) and -37.91% at M12 (p<0.001); DPD-33.4% at M6 (p<0.001) and -33.18% (p<0.001) at M12: NTX -57.08% (p<0.001) at M6 and -55.95% (p<0.001) at M12; OC-11.62% (p=0.05) at M6 and -12.62% at M12 (p=0.06); B-ALP -13.95 % at M6 (p=0.04) and -0.85% at M12 (NS).

Conclusion: A twelve-month intramuscular NE treatment in rheumatic patients under GCs therapy improves lumbar and femoral BMD and mainly reduces the markers of bone resorption.

Publication types

  • Multicenter Study
  • Randomized Controlled Trial

MeSH terms

  • Adolescent
  • Adult
  • Aged
  • Aged, 80 and over
  • Antirheumatic Agents / adverse effects*
  • Biomarkers / blood
  • Bone Density / drug effects
  • Bone Density / physiology
  • Bone Density Conservation Agents / administration & dosage
  • Bone Density Conservation Agents / therapeutic use*
  • Bone Resorption / blood
  • Bone Resorption / drug therapy*
  • Bone Resorption / physiopathology
  • Diphosphonates / administration & dosage
  • Diphosphonates / therapeutic use*
  • Drug Therapy, Combination
  • Female
  • Femur / drug effects
  • Femur / metabolism
  • Glucocorticoids / adverse effects*
  • Humans
  • Injections, Intramuscular
  • Lumbar Vertebrae / drug effects
  • Lumbar Vertebrae / metabolism
  • Male
  • Middle Aged
  • Osteoporosis / chemically induced
  • Osteoporosis / drug therapy
  • Osteoporosis / metabolism
  • Rheumatic Diseases / blood
  • Rheumatic Diseases / complications
  • Rheumatic Diseases / drug therapy*
  • Young Adult

Substances

  • Antirheumatic Agents
  • Biomarkers
  • Bone Density Conservation Agents
  • Diphosphonates
  • Glucocorticoids
  • 6-amino-1-hydroxyhexane-1,1-diphosphonate