Efficacy, safety, and pharmacokinetics of intramuscular hepatitis B immune globulin, Igantibe, for the prophylaxis of viral B hepatitis after liver transplantation

Dig Liver Dis. 2010 Jul;42(7):509-14. doi: 10.1016/j.dld.2009.09.005. Epub 2009 Oct 13.

Abstract

Background: Long-term prophylaxis of hepatitis B virus (HBV) positive liver transplanted subjects with intravenous hepatitis B immunoglobulin (HBIG) is effective, however use of intramuscular HBIG could be as effective with fewer adverse events and lower cost.

Aim: We conducted a prospective, non-randomized, clinical study to assess the efficacy and safety of HBIG from Grifols, Igantibe, for the prophylaxis of HBV reactivation.

Methods: Eighteen adult patients submitted to liver transplantation for HBV-related disease more than 18 months earlier were treated with doses of 2000 I.U. intramuscular Igantibe every 14 days for 6 months.

Results: Mean trough serum HBsAb IgG titers from months 4 to 6 (primary efficacy variable) were protective (>or=150 I.U./L) at each time point. Individual measurements were also protective throughout the study. HBV replication remained negative for all available subjects until study completion. Pharmacokinetic analysis showed a half-life of 27 days and extensive exposure to the study drug. Safety and tolerability of intramuscular Igantibe were good, with only one adverse event.

Conclusion: Standard-dose intramuscular Igantibe administration proved efficacious in post-liver transplantation prophylaxis by attaining protective levels for up to 6 months, was safe and well tolerated. Pharmacokinetic analysis revealed a long half-life and extensive exposure.

Publication types

  • Clinical Trial
  • Multicenter Study

MeSH terms

  • Aged
  • Female
  • Hepatitis B / immunology
  • Hepatitis B / prevention & control*
  • Hepatitis B Antibodies
  • Humans
  • Immunization, Passive*
  • Immunoglobulins / administration & dosage
  • Immunoglobulins / therapeutic use*
  • Immunologic Factors / administration & dosage
  • Immunologic Factors / pharmacokinetics*
  • Injections, Intramuscular
  • Liver Transplantation*
  • Male
  • Middle Aged

Substances

  • Hepatitis B Antibodies
  • Immunoglobulins
  • Immunologic Factors
  • igantibe
  • hepatitis B hyperimmune globulin