Kaposi's sarcoma-associated herpesvirus-encoded viral FLICE inhibitory protein (vFLIP) K13 suppresses CXCR4 expression by upregulating miR-146a

Oncogene. 2010 Mar 25;29(12):1835-44. doi: 10.1038/onc.2009.460. Epub 2009 Dec 21.

Abstract

Kaposi's sarcoma (KS)-associated herpesvirus (KSHV)-encoded viral FLICE inhibitory protein (vFLIP) K13 is a potent activator of the nuclear factor-kappaB (NF-kappaB) pathway. In this study, we show that infection with KHSV and ectopic expression of K13, but not its NF-kappaB-defective mutant, suppressed the expression of CXCR4. Suppression of CXCR4 by KSHV and K13 was associated with upregulated expression of miR-146a, a microRNA that is known to bind to the 3'-untranslated region of CXCR4 mRNA. Reporter studies identified two NF-kappaB sites in the promoter of miR-146a that were essential for its activation by K13. Accordingly, ectopic expression of K13, but not its NF-kappaB-defective mutant or other vFLIPs, strongly stimulated the miR-146a promoter activity, which could be blocked by specific genetic and pharmacological inhibitors of the NF-kappaB pathway. Finally, expression of CXCR4 was downregulated in clinical samples of KS and this was accompanied by an increased expression of miR-146a. Our results show that K13-induced NF-kappaB activity suppresses CXCR4 through upregulation of miR-146a. Downregulation of CXCR4 expression by K13 may contribute to KS development by promoting premature release of KSHV-infected endothelial progenitors into the circulation.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • CASP8 and FADD-Like Apoptosis Regulating Protein / genetics*
  • Down-Regulation
  • Endothelium, Vascular / virology
  • Gene Expression Regulation
  • Genes, Reporter
  • Herpesvirus 8, Human / genetics*
  • Herpesvirus 8, Human / pathogenicity
  • Humans
  • Luciferases / genetics
  • MicroRNAs / genetics*
  • NF-kappa B / genetics
  • Oligonucleotide Array Sequence Analysis
  • Promoter Regions, Genetic
  • Receptors, CXCR4 / genetics*
  • Sarcoma, Kaposi / genetics*
  • Sarcoma, Kaposi / virology
  • Suppression, Genetic
  • Up-Regulation
  • Viral Proteins / genetics

Substances

  • CASP8 and FADD-Like Apoptosis Regulating Protein
  • CXCR4 protein, human
  • MIRN146 microRNA, human
  • MicroRNAs
  • NF-kappa B
  • Receptors, CXCR4
  • Viral Proteins
  • viral FLIP protein, Human herpesvirus 8
  • Luciferases