Activation of the integrin effector kinase focal adhesion kinase in cancer cells is regulated by crosstalk between protein kinase Calpha and the PDZ adapter protein mda-9/Syntenin

Cancer Res. 2010 Feb 15;70(4):1645-55. doi: 10.1158/0008-5472.CAN-09-2447. Epub 2010 Feb 9.

Abstract

Aberrant adhesion signaling pathways in cancer cells underlie their deadly invasive capabilities. The adhesion-related PDZ adapter protein mda-9/syntenin is a positive regulator of cancer cell progression in breast cancer, melanoma, and other human cancers. In this study, we report that mda-9/syntenin mediates adhesion-mediated activation of protein kinase Calpha (PKCalpha) and focal adhesion kinase (FAK) by fibronectin (FN) in human breast cancer and melanoma cells. FN rapidly stimulated the expression of mda-9/syntenin and the activation of PKCalpha prior to activation of FAK. Inhibiting PKCalpha suppressed basal or FN-induced expression of mda-9/syntenin, as well as cell migration and invasion toward FN stimulated by mda-9/syntenin. Several lines of evidence suggested that activation of PKCalpha and expression of mda-9/syntenin were interdependent. First, mda-9/syntenin inhibition suppressed basal or FN-induced phosphorylation of PKCalpha at Thr(638/641), whereas PKCalpha inhibition suppressed basal or FN-induced expression of mda-9/syntenin. Second, inhibiting either mda-9/syntenin or PKCalpha suppressed FN-induced formation of integrin-beta(1)/FAK/c-Src signaling complexes. Third, inhibiting either mda-9/syntenin or PKCalpha suppressed FN-induced phosphorylation of FAK Tyr(397) and c-Src Tyr(416) and the induction of downstream effector signals to p38 and mitogen-activated protein kinase, Cdc42, and NF-kappaB. In summary, our findings offer evidence that mda-9/syntenin acts as a molecular adaptor linking PKCalpha and FAK activation in a pathway of FN adhesion by human breast cancer and melanoma cells.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • CSK Tyrosine-Protein Kinase
  • Cell Adhesion / drug effects
  • Cell Adhesion / genetics
  • Enzyme Activation / drug effects
  • Fibronectins / genetics
  • Fibronectins / physiology
  • Focal Adhesion Protein-Tyrosine Kinases / metabolism*
  • Gene Expression Regulation, Enzymologic / drug effects
  • Gene Expression Regulation, Neoplastic / drug effects
  • Humans
  • Integrin beta1 / metabolism
  • Neoplasms / enzymology
  • Neoplasms / genetics
  • Neoplasms / metabolism*
  • Neoplasms / pathology
  • PDZ Domains / physiology
  • Phosphorylation / drug effects
  • Protein Binding / drug effects
  • Protein Kinase C-alpha / metabolism*
  • Protein Kinase C-alpha / physiology
  • Protein-Tyrosine Kinases / metabolism
  • RNA, Small Interfering / pharmacology
  • Receptor Cross-Talk / physiology
  • Syntenins / antagonists & inhibitors
  • Syntenins / chemistry
  • Syntenins / genetics
  • Syntenins / metabolism*
  • Tumor Cells, Cultured
  • src-Family Kinases

Substances

  • Fibronectins
  • Integrin beta1
  • RNA, Small Interfering
  • SDCBP protein, human
  • Syntenins
  • Protein-Tyrosine Kinases
  • CSK Tyrosine-Protein Kinase
  • Focal Adhesion Protein-Tyrosine Kinases
  • src-Family Kinases
  • CSK protein, human
  • Protein Kinase C-alpha