'TRPing' synaptic ribbon function in the rat pineal gland: neuroendocrine regulation involves the capsaicin receptor TRPV1

Neuroendocrinology. 2010;92(2):133-42. doi: 10.1159/000289765. Epub 2010 Apr 17.

Abstract

Synaptic ribbons (SRs) are presynaptic structures thought to regulate and facilitate multivesicular release. In the pineal gland, they display a circadian rhythm with higher levels at night paralleling melatonin synthesis. To gain more insight into the processes involved and the possible functions of these structures, a series of experiments were conducted in rodents. We studied the regional distribution of a molecular marker of pineal SRs, the kinesin motor KIF3A in the gland. Respective immunoreactivity was abundant in central regions of the gland where sympathetic fibers were less dense, and vice versa, revealing that intercellular communication between adjacent pinealocytes is enhanced under low sympathetic influence. KIF3A was found to be colocalized to the transient receptor potential channel of the vanilloid receptor family, subtype 1 (TRPV1). The TRPV1 agonist capsaicin increased melatonin secretion from perifused pineals in a dose-dependent manner that was blocked by the competitive TRPV1 antagonist capsazepine. No change in free intracellular calcium was observed in response to TRPV1 ligands applied to pinealocytes responding to norepinephrine, bradykinin and/or depolarization. These data clearly indicate that TRPV1 actively regulates pineal gland function.

MeSH terms

  • Animals
  • Bradykinin / physiology
  • Calcium / analysis
  • Capsaicin / analogs & derivatives
  • Capsaicin / pharmacology
  • Kinesins / analysis
  • Kinesins / physiology
  • Melatonin / metabolism
  • Membrane Potentials / physiology
  • Norepinephrine / physiology
  • Pineal Gland / drug effects
  • Pineal Gland / metabolism
  • Pineal Gland / physiology*
  • Rats
  • Rats, Sprague-Dawley
  • Synapses / physiology*
  • TRPV Cation Channels / physiology*

Substances

  • Kif3a protein, rat
  • TRPV Cation Channels
  • Trpv1 protein, rat
  • Kinesins
  • Melatonin
  • capsazepine
  • Capsaicin
  • Bradykinin
  • Calcium
  • Norepinephrine