The PD-1/PD-L1 axis modulates the natural killer cell versus multiple myeloma effect: a therapeutic target for CT-011, a novel monoclonal anti-PD-1 antibody

Blood. 2010 Sep 30;116(13):2286-94. doi: 10.1182/blood-2010-02-271874. Epub 2010 May 11.

Abstract

T-cell expression of programmed death receptor-1 (PD-1) down-regulates the immune response against malignancy by interacting with cognate ligands (eg, PD-L1) on tumor cells; however, little is known regarding PD-1 and natural killer (NK) cells. NK cells exert cytotoxicity against multiple myeloma (MM), an effect enhanced through novel therapies. We show that NK cells from MM patients express PD-1 whereas normal NK cells do not and confirm PD-L1 on primary MM cells. Engagement of PD-1 with PD-L1 should down-modulate the NK-cell versus MM effect. We demonstrate that CT-011, a novel anti-PD-1 antibody, enhances human NK-cell function against autologous, primary MM cells, seemingly through effects on NK-cell trafficking, immune complex formation with MM cells, and cytotoxicity specifically toward PD-L1(+) MM tumor cells but not normal cells. We show that lenalidomide down-regulates PD-L1 on primary MM cells and may augment CT-011's enhancement of NK-cell function against MM. We demonstrate a role for the PD-1/PD-L1 signaling axis in the NK-cell immune response against MM and a role for CT-011 in enhancing the NK-cell versus MM effect. A phase 2 clinical trial of CT-011 in combination with lenalidomide for patients with MM should be considered.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antibodies, Monoclonal / administration & dosage
  • Antibodies, Monoclonal / therapeutic use*
  • Antigen-Antibody Complex / metabolism
  • Antigens, CD / metabolism*
  • Antineoplastic Agents / administration & dosage
  • Apoptosis Regulatory Proteins / metabolism*
  • B7-H1 Antigen
  • Cell Line, Tumor
  • Chemokine CXCL12 / metabolism
  • Cytotoxicity, Immunologic
  • Down-Regulation / drug effects
  • Humans
  • In Vitro Techniques
  • Interferon-gamma / biosynthesis
  • K562 Cells
  • Killer Cells, Natural / immunology*
  • Lenalidomide
  • Multiple Myeloma / immunology*
  • Multiple Myeloma / therapy*
  • Programmed Cell Death 1 Receptor
  • Receptors, CXCR4 / metabolism
  • Signal Transduction / immunology
  • Thalidomide / administration & dosage
  • Thalidomide / analogs & derivatives

Substances

  • Antibodies, Monoclonal
  • Antigen-Antibody Complex
  • Antigens, CD
  • Antineoplastic Agents
  • Apoptosis Regulatory Proteins
  • B7-H1 Antigen
  • CD274 protein, human
  • CXCL12 protein, human
  • CXCR4 protein, human
  • Chemokine CXCL12
  • PDCD1 protein, human
  • Programmed Cell Death 1 Receptor
  • Receptors, CXCR4
  • Thalidomide
  • Interferon-gamma
  • Lenalidomide