The effect of donepezil treatment on cardiovascular mortality

Clin Pharmacol Ther. 2010 Sep;88(3):335-8. doi: 10.1038/clpt.2010.98. Epub 2010 Jul 21.

Abstract

The acetylcholinesterase inhibitor donepezil hydrochloride improves cognitive function in patients with Alzheimer's disease and vascular dementia. Given acetylcholine's important actions on the heart, we undertook a retrospective cohort investigation to assess whether donepezil usage affects cardiovascular mortality. In patients treated with donepezil, hazard ratios for total and cardiovascular mortality were 0.68 (P = 0.045, 95% confidence interval 0.46-0.99) and 0.54 (P = 0.042, 95% confidence interval 0.30-0.98), respectively. The apparent survival benefit in donepezil-treated patients should not be overinterpreted. Prospective clinical trials are warranted.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Aged
  • Aged, 80 and over
  • Alzheimer Disease / complications
  • Alzheimer Disease / drug therapy*
  • Cardiovascular Diseases / complications
  • Cardiovascular Diseases / drug therapy*
  • Cardiovascular Diseases / mortality
  • Cholinesterase Inhibitors / adverse effects
  • Cholinesterase Inhibitors / pharmacology*
  • Cholinesterase Inhibitors / therapeutic use
  • Cohort Studies
  • Dementia, Vascular / complications
  • Dementia, Vascular / drug therapy*
  • Donepezil
  • Female
  • Follow-Up Studies
  • Humans
  • Indans / adverse effects
  • Indans / pharmacology*
  • Indans / therapeutic use
  • Male
  • Nootropic Agents / adverse effects
  • Nootropic Agents / pharmacology
  • Nootropic Agents / therapeutic use
  • Piperidines / adverse effects
  • Piperidines / pharmacology*
  • Piperidines / therapeutic use
  • Proportional Hazards Models
  • Retrospective Studies

Substances

  • Cholinesterase Inhibitors
  • Indans
  • Nootropic Agents
  • Piperidines
  • Donepezil