Rosiglitazone and vascular injury in hypercholesterolemic rabbits: neointimal formation assessment

Arq Bras Cardiol. 2010 Sep;95(3):283-8. doi: 10.1590/s0066-782x2010005000101. Epub 2010 Jul 30.

Abstract

Background: Rosiglitazone has been the focus of extensive discussion.

Objective: To evaluate the effects of rosiglitazone on iliac arteries, both at the injury site and the contralateral artery, of hypercholesterolemic rabbits undergoing balloon catheter injury.

Methods: White male rabbits were fed a hypercholesterolemic diet by oral gavage for 6 weeks and divided into two groups as follows: rosiglitazone group (14 rabbits treated with rosiglitazone during 6 weeks) and the control group (18 rabbits without rosiglitazone). Animals underwent balloon catheter injury of the right iliac artery on the 14th day.

Results: In the contralateral iliac artery, there was no significant difference in the intima/media layer area ratio (IMR) between the control and rosiglitazone groups. Rosiglitazone did not reduce the probability of type I, II, or III lesions (72.73% vs 92.31%; p=0.30) and type IV or V lesions (27.27% vs 7.69%; p=0.30). As for the homolateral iliac artery, the intimal area was significantly lower in the rosiglitazone group, as compared to the control group (p = 0.024). The luminal layer area was higher in the rosiglitazone group vs. the control group (p < 0.0001). There was a significant reduction of 65% in the IMR in the rosiglitazone group vs the control group (p = 0.021). None of the histological criteria for type I-V atherosclerotic lesions (American Heart Association) were found in the homolateral iliac artery.

Conclusion: These findings demonstrate that rosiglitazone given for 6 weeks prevents atherogenesis at the injury site, but not in a vessel distant from the injury site.

MeSH terms

  • Animals
  • Anti-Inflammatory Agents / pharmacology
  • Atherosclerosis / prevention & control*
  • Disease Models, Animal
  • Hypercholesterolemia / complications*
  • Hypercholesterolemia / metabolism
  • Iliac Artery / drug effects*
  • Iliac Artery / injuries
  • Iliac Artery / metabolism
  • Iliac Artery / pathology
  • Male
  • Neointima / etiology*
  • Neointima / metabolism
  • Rabbits
  • Random Allocation
  • Rosiglitazone
  • Thiazolidinediones / pharmacology*

Substances

  • Anti-Inflammatory Agents
  • Thiazolidinediones
  • Rosiglitazone