Effect of high pH mobile phase on the sensitivity of multiple drugs by LC positive electrospray ionization MS/MS

Bioanalysis. 2009 Nov;1(8):1419-30. doi: 10.4155/bio.09.133.

Abstract

Background: In this study, the postcolumn addition approach was used to evaluate the impact of high pH modifiers on the sensitivity of 25 compounds by LC-MS/MS under positive ESI (ESI+).

Results: None of the compounds were significantly suppressed by the use of high pH modifiers. Most of them showed a signal enhancement by at least twofold compared with acidic modifiers. The sensitivity gained under high pH mobile phase was used to develop a bioassay for the quantification of candesartan. The use of high pH mobile phase allowed for fast sample preparation that would have been impossible under typical low pH chromatography.

Conclusion: We have shown that high pH modifiers are sufficient to induce a signal enhancement for the majority of compounds detected under LC-ESI+-MS/MS.

MeSH terms

  • Analytic Sample Preparation Methods
  • Animals
  • Benzimidazoles / blood
  • Benzimidazoles / metabolism
  • Biphenyl Compounds
  • Chromatography, Liquid / methods*
  • Humans
  • Hydrogen-Ion Concentration
  • Limit of Detection
  • Pharmaceutical Preparations / blood*
  • Pharmaceutical Preparations / metabolism
  • Sensitivity and Specificity
  • Spectrometry, Mass, Electrospray Ionization / methods*
  • Tandem Mass Spectrometry / methods
  • Tetrazoles / blood
  • Tetrazoles / metabolism

Substances

  • Benzimidazoles
  • Biphenyl Compounds
  • Pharmaceutical Preparations
  • Tetrazoles
  • candesartan