The effect of exemestane, anastrozole, and tamoxifen on lipid profiles in Japanese postmenopausal early breast cancer patients: final results of National Surgical Adjuvant Study BC 04, the TEAM Japan sub-study

Ann Oncol. 2011 Aug;22(8):1777-82. doi: 10.1093/annonc/mdq707. Epub 2011 Feb 1.

Abstract

Background: In this Tamoxifen Exemestane Adjuvant Multinational Japan sub-study, we evaluated the time course of changes in serum lipids in postmenopausal women with hormone-sensitive early breast cancer treated with exemestane, anastrozole, or tamoxifen for postoperative adjuvant therapy.

Patients and methods: A total of 154 breast cancer patients were assigned to receive exemestane, anastrozole, or tamoxifen in this randomized open-label study. Serum lipid parameters including triglyceride (TG), total cholesterol (TC), high-density lipoprotein cholesterol (HDL-C), and low-density lipoprotein cholesterol (LDL-C) were measured during 1 year of treatment.

Results: TC and LDL-C rapidly decreased in patients treated with tamoxifen at 3 months. Compared with anastrozole and exemestane patients, TC and LDL-C were significantly lower at all assessment time points in tamoxifen patients (P < 0.05). TG increased in tamoxifen patients; it was significantly higher compared with exemestane patients at all assessment time points (P < 0.05). HDL-C slightly decreased in exemestane patients; it was significantly lower compared with anastrozole patients at 3 months and 1 year (P = 0.0179 and 0.0013, respectively).

Conclusion: Changes of lipid profiles in Japanese postmenopausal women treated with tamoxifen were relatively favorable, while exemestane and anastrozole had no clinically significant effect on the serum lipids.

Publication types

  • Multicenter Study
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aged
  • Aged, 80 and over
  • Anastrozole
  • Androstadienes / therapeutic use*
  • Aromatase Inhibitors / therapeutic use
  • Breast Neoplasms / blood*
  • Breast Neoplasms / drug therapy*
  • Breast Neoplasms / pathology
  • Chemotherapy, Adjuvant
  • Cholesterol / blood
  • Cholesterol, HDL / blood
  • Cholesterol, LDL / blood
  • Female
  • Humans
  • Japan
  • Lipids / blood*
  • Middle Aged
  • Neoplasm Staging
  • Neoplasms, Hormone-Dependent / blood*
  • Neoplasms, Hormone-Dependent / drug therapy*
  • Neoplasms, Hormone-Dependent / pathology
  • Nitriles / therapeutic use*
  • Postmenopause / blood
  • Tamoxifen / therapeutic use*
  • Triazoles / therapeutic use*
  • Triglycerides / blood

Substances

  • Androstadienes
  • Aromatase Inhibitors
  • Cholesterol, HDL
  • Cholesterol, LDL
  • Lipids
  • Nitriles
  • Triazoles
  • Triglycerides
  • Tamoxifen
  • Anastrozole
  • Cholesterol
  • exemestane