DUSP13B/TMDP inhibits stress-activated MAPKs and suppresses AP-1-dependent gene expression

Mol Cell Biochem. 2011 Jun;352(1-2):155-62. doi: 10.1007/s11010-011-0749-x. Epub 2011 Mar 1.

Abstract

The dual-specificity phosphatase (DUSP) 13 gene encodes two atypical DUSPs, DUSP13B/TMDP and DUSP13A/MDSP using alternative exons. DUSP13B protein is most highly expressed in testis, particularly in spermatocytes and round spermatids of the seminiferous tubules, while that of DUSP13A is restricted to skeletal muscle. Here, we show that DUSP13B inactivated MAPK activation in the order of selectivity, JNK = p38>ERK in cells, while DUSP13A did not show MAPK phosphatase activity. Reporter gene analysis showed that DUSP13B had significant inhibitory effect on AP-1-dependent gene expression, but DUSP13A did not. To our knowledge, DUSP13B is the first identified testis-specific phosphatase that inhibits stress-activated MAPKs. These data suggest an important role for DUSP13B in protection from external stress during spermatogenesis.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cell Line
  • Dual-Specificity Phosphatases / physiology*
  • Enzyme Activation
  • Exons
  • Gene Expression Regulation / physiology*
  • Humans
  • Mitogen-Activated Protein Kinases / antagonists & inhibitors
  • Mitogen-Activated Protein Kinases / metabolism*
  • Protein Kinase Inhibitors / pharmacology
  • Transcription Factor AP-1 / physiology*

Substances

  • Protein Kinase Inhibitors
  • Transcription Factor AP-1
  • Mitogen-Activated Protein Kinases
  • DUSP13 protein, human
  • Dual-Specificity Phosphatases