Monoclonal anti-HMGB1 (high mobility group box chromosomal protein 1) antibody protection in two experimental arthritis models

Mol Med. 2011 Sep-Oct;17(9-10):1039-44. doi: 10.2119/molmed.2010.00264. Epub 2011 Jun 7.

Abstract

High mobility group box chromosomal protein 1 (HMGB1) is a DNA-binding nuclear protein that can be released from dying cells and activated myeloid cells. Extracellularly, HMGB1 promotes inflammation. Experimental studies demonstrate HMGB1 to be a pathogenic factor in many inflammatory conditions including arthritis. HMGB1-blocking therapies in arthritis models alleviate disease and confer significant protection against cartilage and bone destruction. So far, the most successful HMGB1-targeted therapies have been demonstrated with HMGB1-specific polyclonal antibodies and with recombinant A box protein, a fragment of HMGB1. The present study is the first to evaluate the potential of a monoclonal anti-HMGB1 antibody (2G7, mouse IgG2b) to ameliorate arthritis. Effects of repeated injections of this antibody have now been studied in two conceptually different models of arthritis: collagen type II-induced arthritis (CIA) in DBA/1 mice and in a spontaneous arthritis disease in mice with combined deficiencies for genes encoding for the enzyme DNase type II and interferon type I receptors. These mice are unable to degrade phagocytozed DNA in macrophages and develop chronic, destructive polyarthritis. Therapeutic intervention in CIA and prophylactic administration of anti-HMGB1 monoclonal antibody (mAb) in the spontaneous arthritis model significantly ameliorated the clinical courses. Anti-HMGB1 mAb therapy also partially prevented joint destruction, as demonstrated by histological examination. The beneficial antiarthritic effects by the anti-HMGB1 mAb in two diverse models of arthritis represent additional proof-of-concept, indicating that HMGB1 may be a valid target molecule to consider for development of future clinical therapy.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Ankle Joint / drug effects
  • Ankle Joint / pathology
  • Antibodies, Monoclonal / immunology
  • Antibodies, Monoclonal / pharmacology*
  • Arthritis, Experimental / chemically induced
  • Arthritis, Experimental / pathology
  • Arthritis, Experimental / prevention & control*
  • Collagen Type II
  • Endodeoxyribonucleases / deficiency
  • Endodeoxyribonucleases / genetics
  • Female
  • HMGB1 Protein / antagonists & inhibitors*
  • HMGB1 Protein / immunology
  • Joints / drug effects*
  • Joints / pathology
  • Male
  • Metacarpophalangeal Joint / drug effects
  • Metacarpophalangeal Joint / pathology
  • Metatarsophalangeal Joint / drug effects
  • Metatarsophalangeal Joint / pathology
  • Mice
  • Mice, Inbred DBA
  • Mice, Knockout
  • Receptor, Interferon alpha-beta / deficiency
  • Receptor, Interferon alpha-beta / genetics
  • Severity of Illness Index
  • Time Factors

Substances

  • Antibodies, Monoclonal
  • Collagen Type II
  • HMGB1 Protein
  • Receptor, Interferon alpha-beta
  • Endodeoxyribonucleases
  • deoxyribonuclease II