Montelukast was inefficient in maintaining steroid-induced remission in adult eosinophilic esophagitis

Dig Dis Sci. 2011 Dec;56(12):3551-8. doi: 10.1007/s10620-011-1775-y. Epub 2011 Jun 15.

Abstract

Background and aims: Leukotriene D4 is produced by and functions as a chemotactic factor for eosinophils. Eosinophilic esophagitis (EoE) is characterized by esophageal eosinophilic infiltration, determining structural changes and dismotility symptoms. Montelukast, a selective leukotriene D4 receptor antagonist, has gained increasing consideration as a therapeutic agent for EoE. However, limited available information has shown that montelukast is not effective in reducing eosinophilic infiltration. Our paper aims at evaluating whether montelukast could be consider as a steroid-sparing therapy by assessing its efficacy in maintaining both clinical and histopathological remission achieved after topical corticosteroids in adult EoE patients.

Methods: Eleven consecutively diagnosed adult EoE patients were prospectively studied. Esophageal biopsies were obtained before and after a 6-month treatment with fluticasone propionate 400 μg/twice a day. Immediately after that, montelukast 10 mg/day was instituted. A new endoscopy was foreseen after a new 3-month period, or as soon as the patients presented esophageal symptoms. Symptoms were assessed by using a questionnaire before and after fluticasone propionate treatment and after montelukast therapy.

Results: Eosinophils density into the esophageal epithelium and lamina propria was significantly reduced after a 6-month treatment with topical steroids (P = 0.003) and increased to levels similar to baseline level into the first 3 months after treatment with montelukast. Baseline symptom scores significantly decreased after treatment with topical steroids (P = 0.003) and increased again after montelukast therapy, but baseline levels improved.

Conclusions: Montelukast was not efficient in maintaining the histopathological or clinical response achieved by topical steroids in adult EoE patients.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acetates / administration & dosage
  • Acetates / therapeutic use*
  • Adult
  • Androstadienes / administration & dosage
  • Androstadienes / therapeutic use*
  • Anti-Inflammatory Agents / administration & dosage
  • Anti-Inflammatory Agents / therapeutic use
  • Biopsy
  • Cyclopropanes
  • Dose-Response Relationship, Drug
  • Drug Therapy, Combination
  • Endoscopy, Gastrointestinal
  • Eosinophilic Esophagitis / drug therapy*
  • Eosinophilic Esophagitis / metabolism
  • Eosinophilic Esophagitis / pathology
  • Female
  • Fluticasone
  • Follow-Up Studies
  • Humans
  • Leukotriene Antagonists / administration & dosage
  • Leukotriene Antagonists / therapeutic use*
  • Male
  • Middle Aged
  • Patient Satisfaction
  • Prospective Studies
  • Quinolines / administration & dosage
  • Quinolines / therapeutic use*
  • Remission Induction / methods
  • Sulfides
  • Surveys and Questionnaires
  • Treatment Outcome
  • Young Adult

Substances

  • Acetates
  • Androstadienes
  • Anti-Inflammatory Agents
  • Cyclopropanes
  • Leukotriene Antagonists
  • Quinolines
  • Sulfides
  • Fluticasone
  • montelukast