ADP-ribosylarginine hydrolase regulates cell proliferation and tumorigenesis

Cancer Res. 2011 Aug 1;71(15):5327-35. doi: 10.1158/0008-5472.CAN-10-0733. Epub 2011 Jun 22.

Abstract

Protein ADP-ribosylation is a reversible posttranslational modification of uncertain significance in cancer. In this study, we evaluated the consequences for cancer susceptibility in the mouse of a genetic deletion of the enzyme responsible for removing mono-ADP-ribose moieties from arginines in cellular proteins. Specifically, we analyzed cancer susceptibility in animals lacking the ADP-ribosylarginine hydrolase (ARH1) that cleaves the ADP ribose-protein bond. ARH1(-/-) cells or ARH1(-/-) cells overexpressing an inactive mutant ARH1 protein (ARH1(-/-)+dm) had higher proliferation rates than either wild-type ARH1(+/+) cells or ARH1(-/-) cells engineered to express the wild-type ARH1 enzyme. More significantly, ARH1(-/-) and ARH1(+/-) mice spontaneously developed lymphomas, adenocarcinomas, and metastases more frequently than wild-type ARH1(+/+) mice. In ARH1(+/-) mice, we documented in all arising tumors mutation of the remaining wild-type allele (or loss of heterozygosity), illustrating the strict correlation that existed between tumor formation and absence of ARH1 gene function. Our findings show that proper control of protein ADP-ribosylation levels affected by ARH1 is essential for cancer suppression.

Publication types

  • Research Support, N.I.H., Intramural

MeSH terms

  • Adenosine Diphosphate Ribose / analogs & derivatives
  • Adenosine Diphosphate Ribose / metabolism
  • Animals
  • Cell Division
  • Cell Transformation, Neoplastic / genetics*
  • Cell Transformation, Neoplastic / metabolism
  • Female
  • Genetic Predisposition to Disease
  • Genotype
  • Loss of Heterozygosity
  • Mice
  • Mice, Inbred BALB C
  • Mice, Inbred C57BL
  • Mice, Knockout
  • Mice, Nude
  • N-Glycosyl Hydrolases / deficiency
  • N-Glycosyl Hydrolases / genetics
  • N-Glycosyl Hydrolases / physiology*
  • Neoplasm Metastasis / genetics*
  • Neoplasm Proteins / physiology*
  • Neoplasms, Experimental / enzymology*
  • Neoplasms, Experimental / genetics
  • Protein Processing, Post-Translational
  • Tumor Stem Cell Assay

Substances

  • Neoplasm Proteins
  • Adenosine Diphosphate Ribose
  • ADP-ribosylarginine
  • N-Glycosyl Hydrolases
  • ADP-ribosylarginine hydrolase