p300-Dependent ATF5 acetylation is essential for Egr-1 gene activation and cell proliferation and survival

Mol Cell Biol. 2011 Sep;31(18):3906-16. doi: 10.1128/MCB.05887-11. Epub 2011 Jul 26.

Abstract

ATF5 has been shown to be a critical regulator of cell proliferation and survival; however, the underlying mechanism remains largely unknown. We demonstrate here that ATF5 interacts with the transcriptional coactivator p300, which acetylates ATF5 at lysine-29 (K29), which in turn enhances the interaction between ATF5 and p300 and binding of the ATF5/p300 complex to the ATF5 response element (ARE) region of the Egr-1 promoter. ARE-bound ATF5/p300 acetylates lysine-14 (K14) of nucleosomal histone H3 at both the ARE and serum response element (SRE) of the Egr-1 promoter, which facilitates binding of extracellular signal-regulated kinase (ERK)-phosphorylated Elk-1 to the SRE, activating the Egr-1 promoter. Interference of p300-dependent acetylation of ATF5 or nucleosomal histone H3 or blockade of ERK-dependent Elk-1 phosphorylation abrogates ATF5-dependent Egr-1 activation and cell proliferation and survival. These findings assign a central role for the ATF5/p300 complex in ATF5 function and suggest that coordinated actions by ATF5, p300, Elk-1, and ERK/mitogen-activated protein kinase (MAPK) are essential for ATF5-dependent Egr-1 activation and cell proliferation and survival.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Acetylation
  • Activating Transcription Factors / metabolism*
  • Cell Line, Tumor
  • Cell Proliferation*
  • Cell Survival*
  • DNA-Binding Proteins / metabolism
  • E1A-Associated p300 Protein / metabolism*
  • Early Growth Response Protein 1 / biosynthesis
  • Early Growth Response Protein 1 / genetics*
  • Early Growth Response Protein 1 / metabolism
  • Extracellular Signal-Regulated MAP Kinases / genetics
  • Extracellular Signal-Regulated MAP Kinases / metabolism
  • HEK293 Cells
  • Histones / metabolism
  • Humans
  • Promoter Regions, Genetic
  • RNA Interference
  • RNA, Small Interfering
  • Response Elements*
  • Reverse Transcriptase Polymerase Chain Reaction
  • Signal Transduction / genetics
  • Transcription Factors / metabolism

Substances

  • ATF5 protein, human
  • Activating Transcription Factors
  • DNA-Binding Proteins
  • Early Growth Response Protein 1
  • Histones
  • RNA, Small Interfering
  • SRE protein, human
  • Transcription Factors
  • E1A-Associated p300 Protein
  • EP300 protein, human
  • Extracellular Signal-Regulated MAP Kinases