Treatment with valacyclovir, famciclovir, or antiretrovirals reduces human herpesvirus-8 replication in HIV-1 seropositive men

J Med Virol. 2011 Oct;83(10):1696-703. doi: 10.1002/jmv.22194.

Abstract

Human herpesvirus-8 (HHV-8) replication is a key factor in Kaposi sarcoma, primary effusion lymphoma, and Castleman disease pathogenesis. In vitro data suggest that antivirals inhibit HHV-8 replication, but little data exist in humans. Daily oropharyngeal swabs were analyzed from HIV/HHV-8 dually infected men enrolled in three previous clinical trials of valacyclovir and famciclovir for HIV-1 and/or HSV-2 suppression. Fifty-eight participants contributed 6,036 swabs. HHV-8 was detected in 1,128 (19%) of 6,036 swabs, including 618 (21%) of 2,992 on placebo, 323 (15%) of 2,221 on valacyclovir, and 187 (23%) of 823 on famciclovir. After adjusting for baseline HIV viral load and highly active antiretroviral therapy (HAART) use, an 18% reduction in HHV-8 shedding frequency (IRR 0.822; P = 0.011) was found in participants on valacyclovir and a 30% reduction (IRR 0.700; P < 0.001) on famciclovir. HAART was associated with an 89% (IRR 0.129; P = 0.048) reduction in HHV-8-shedding. Neither antiviral nor antiretroviral therapy was associated with decreased HHV-8 quantity. Valacyclovir and famciclovir were associated with modest but significant reductions in HHV-8 oropharyngeal shedding frequency. In contrast, HAART was a potent inhibitor of HHV-8 replication. Studies of whether antiviral therapy in combination with ART will prevent HHV-8-associated disease appear warranted.

Publication types

  • Clinical Trial
  • Randomized Controlled Trial
  • Research Support, N.I.H., Extramural

MeSH terms

  • 2-Aminopurine / administration & dosage
  • 2-Aminopurine / analogs & derivatives*
  • 2-Aminopurine / pharmacology
  • 2-Aminopurine / therapeutic use
  • AIDS-Related Opportunistic Infections / drug therapy*
  • AIDS-Related Opportunistic Infections / virology
  • Acyclovir / administration & dosage
  • Acyclovir / analogs & derivatives*
  • Acyclovir / pharmacology
  • Acyclovir / therapeutic use
  • Adult
  • Antiretroviral Therapy, Highly Active*
  • Antiviral Agents / administration & dosage
  • Antiviral Agents / pharmacology
  • Antiviral Agents / therapeutic use*
  • Famciclovir
  • HIV-1 / immunology
  • HIV-1 / isolation & purification
  • Herpesviridae Infections / drug therapy*
  • Herpesviridae Infections / virology
  • Herpesvirus 8, Human / drug effects*
  • Herpesvirus 8, Human / isolation & purification
  • Herpesvirus 8, Human / physiology
  • Humans
  • Male
  • Middle Aged
  • Oropharynx / virology
  • Valacyclovir
  • Valine / administration & dosage
  • Valine / analogs & derivatives*
  • Valine / pharmacology
  • Valine / therapeutic use
  • Viral Load
  • Virus Replication / drug effects

Substances

  • Antiviral Agents
  • 2-Aminopurine
  • Valine
  • Valacyclovir
  • Famciclovir
  • Acyclovir