The involvement of the HO-1 pathway in the anti-inflammatory action of a sulfated polysaccharide isolated from the red seaweed Gracilaria birdiae

Inflamm Res. 2011 Dec;60(12):1121-30. doi: 10.1007/s00011-011-0376-8. Epub 2011 Aug 31.

Abstract

Objectives: The aim of this study was to investigate the involvement of the hemoxigenase-1 (HO-1) pathway in the anti-inflammatory action of a sulfated polysaccharide from the red seaweed Gracilaria birdiae (SP-Gb).

Methods: SP-Gb (5, 10 and 20 mg/kg) was administered to Wistar rats in a peritonitis model using carrageenan or a paw edema model using carrageenan or dextran. To analyze the involvement of HO-1 in the anti-inflammatory activity of SP-Gb, the animals were pretreated subcutaneously with a specific HO-1 inhibitor (ZnPP IX). To evaluate the systemic effects, SP-Gb (10 mg/kg) was administered to mice intraperitoneally before waiting for 48 h or for 14 days.

Results: SP-Gb (10 mg/kg) caused an anti-inflammatory effect that was evidenced by a decrease in leukocytes in the peritoneal cavity. SP-Gb also reduced the paw edema induced by carrageenan and inhibited the paw edema induced by dextran in the first half-hour. After being inhibited by ZnPP IX, the anti-inflammatory effect of SP-Gb on carrageenan-induced rat paw edema was not observed. SP-Gb did not cause mortality or significant changes in the biochemical, hematological and histopathological parameters.

Conclusion: SP-Gb may be used as a tool for further investigations into the inflammatory processes associated with the hemoxigenase-1 pathway.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Anti-Inflammatory Agents / isolation & purification
  • Anti-Inflammatory Agents / pharmacology*
  • Anti-Inflammatory Agents / therapeutic use
  • Carrageenan
  • Dextrans
  • Edema / chemically induced
  • Edema / drug therapy
  • Edema / immunology*
  • Enzyme Inhibitors / pharmacology
  • Gracilaria / chemistry*
  • Heme Oxygenase-1 / antagonists & inhibitors
  • Heme Oxygenase-1 / immunology*
  • Leukocyte Count
  • Male
  • Mice
  • Peritonitis / chemically induced
  • Peritonitis / drug therapy
  • Peritonitis / immunology*
  • Peroxidase / metabolism
  • Polysaccharides / isolation & purification
  • Polysaccharides / pharmacology*
  • Polysaccharides / therapeutic use
  • Protoporphyrins / pharmacology
  • Rats
  • Rats, Wistar

Substances

  • Anti-Inflammatory Agents
  • Dextrans
  • Enzyme Inhibitors
  • Polysaccharides
  • Protoporphyrins
  • zinc protoporphyrin
  • Carrageenan
  • Peroxidase
  • Heme Oxygenase-1