Treatment with octreotide does not reduce tumor uptake of (68)Ga-DOTATATE as measured by PET/CT in patients with neuroendocrine tumors

J Nucl Med. 2011 Nov;52(11):1679-83. doi: 10.2967/jnumed.111.089276. Epub 2011 Oct 5.

Abstract

We hypothesized that (68)Ga-DOTATATE uptake of neuroendocrine tumors is sensitive to therapy with a nonradioactive somatostatin analog.

Methods: (68)Ga-DOTATATE PET/CT was used to examine 105 patients, 35 of whom had been pretreated with long-acting octreotide. The maximum standardized uptake value (SUV(max)) of target tissues, as well as metastases, was compared between the groups of patients with (group 1) and without (group 2) octreotide treatment.

Results: The SUV(max) of the spleen and liver was significantly lower in group 1 than in group 2 (both P < 0.001). There were no significant group differences in SUV(max) for primary tumors (28.6 ± 6.8 vs. 32.9 ± 31.5) or metastases in the liver (27.2 ± 14.8 vs. 25.7 ± 10.7), lymph nodes (41.4 ± 19.5 vs. 25.0 ± 6.3), or skeleton (39.5 ± 22.0 vs. 15.4 ± 7.8). In 9 patients available for intraindividual comparison, tumor uptake was unaffected by treatment with somatostatin analogs (21.7 vs. 20.6; P = 0.93).

Conclusion: Treatment with a long-acting somatostatin analog did not significantly reduce (68)Ga-DOTATATE binding in neuroendocrine tumors but tended to improve the tumor-to-background ratio.

Publication types

  • Clinical Trial

MeSH terms

  • Adult
  • Aged
  • Aged, 80 and over
  • Biological Transport / drug effects
  • Female
  • Humans
  • Male
  • Middle Aged
  • Multimodal Imaging*
  • Neoplasm Metastasis
  • Neuroendocrine Tumors / diagnostic imaging*
  • Neuroendocrine Tumors / drug therapy
  • Neuroendocrine Tumors / metabolism*
  • Neuroendocrine Tumors / pathology
  • Octreotide / pharmacology*
  • Octreotide / therapeutic use
  • Organometallic Compounds / metabolism*
  • Positron-Emission Tomography*
  • Tomography, X-Ray Computed*
  • Young Adult

Substances

  • Organometallic Compounds
  • gallium Ga 68 dotatate
  • Octreotide