Carbon monoxide induced PPARγ SUMOylation and UCP2 block inflammatory gene expression in macrophages

PLoS One. 2011;6(10):e26376. doi: 10.1371/journal.pone.0026376. Epub 2011 Oct 25.

Abstract

Carbon monoxide (CO) dampens pro-inflammatory responses in a peroxisome proliferator-activated receptor-γ (PPARγ) and p38 mitogen-activated protein kinase (MAPK) dependent manner. Previously, we demonstrated that CO inhibits lipopolysaccharide (LPS)-induced expression of the proinflammatory early growth response-1 (Egr-1) transcription factor in macrophages via activation of PPARγ. Here, we further characterize the molecular mechanisms by which CO modulates the activity of PPARγ and Egr-1 repression. We demonstrate that CO enhances SUMOylation of PPARγ which we find was attributed to mitochondrial ROS generation. Ectopic expression of a SUMOylation-defective PPARγ-K365R mutant partially abolished CO-mediated suppression of LPS-induced Egr-1 promoter activity. Expression of a PPARγ-K77R mutant did not impair the effect of CO. In addition to PPARγ SUMOylation, CO-activated p38 MAPK was responsible for Egr-1 repression. Blocking both CO-induced PPARγ SUMOylation and p38 activation, completely reversed the effects of CO on inflammatory gene expression. In primary macrophages isolated form C57/BL6 male mice, we identify mitochondrial ROS formation by CO as the upstream trigger for the observed effects on Egr-1 in part through uncoupling protein 2 (UCP2). Macrophages derived from bone marrow isolated from Ucp2 gene Knock-Out C57/BL6 mice (Ucp2(-/-)), produced significantly less ROS with CO exposure versus wild-type macrophages. Moreover, absence of UCP2 resulted in a complete loss of CO mediated Egr-1 repression. Collectively, these results indentify p38 activation, PPARγ-SUMOylation and ROS formation via UCP2 as a cooperative system by which CO impacts the inflammatory response.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Animals
  • Carbon Monoxide / pharmacology*
  • Early Growth Response Protein 1 / metabolism
  • Gene Expression / drug effects
  • Inflammation / chemically induced*
  • Inflammation / genetics
  • Ion Channels / physiology*
  • Macrophages / metabolism*
  • Male
  • Mice
  • Mitochondrial Proteins / physiology*
  • PPAR gamma / metabolism*
  • Reactive Oxygen Species / metabolism
  • Sumoylation / drug effects*
  • Uncoupling Protein 2
  • p38 Mitogen-Activated Protein Kinases / metabolism

Substances

  • Early Growth Response Protein 1
  • Ion Channels
  • Mitochondrial Proteins
  • PPAR gamma
  • Reactive Oxygen Species
  • Ucp2 protein, mouse
  • Uncoupling Protein 2
  • Carbon Monoxide
  • p38 Mitogen-Activated Protein Kinases