Conserved molecular interactions within the HBO1 acetyltransferase complexes regulate cell proliferation

Mol Cell Biol. 2012 Feb;32(3):689-703. doi: 10.1128/MCB.06455-11. Epub 2011 Dec 5.

Abstract

Acetyltransferase complexes of the MYST family with distinct substrate specificities and functions maintain a conserved association with different ING tumor suppressor proteins. ING complexes containing the HBO1 acetylase are a major source of histone H3 and H4 acetylation in vivo and play critical roles in gene regulation and DNA replication. Here, our molecular dissection of HBO1/ING complexes unravels the protein domains required for their assembly and function. Multiple PHD finger domains present in different subunits bind the histone H3 N-terminal tail with a distinct specificity toward lysine 4 methylation status. We show that natively regulated association of the ING4/5 PHD domain with HBO1-JADE determines the growth inhibitory function of the complex, linked to its tumor suppressor activity. Functional genomic analyses indicate that the p53 pathway is a main target of the complex, at least in part through direct transcription regulation at the initiation site of p21/CDKN1A. These results demonstrate the importance of ING association with MYST acetyltransferases in controlling cell proliferation, a regulated link that accounts for the reported tumor suppressor activities of these complexes.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Cell Line
  • Cell Proliferation*
  • Histone Acetyltransferases / chemistry
  • Histone Acetyltransferases / metabolism*
  • Histones / chemistry
  • Histones / metabolism
  • Humans
  • Protein Structure, Tertiary
  • Tumor Suppressor Proteins / chemistry
  • Tumor Suppressor Proteins / metabolism
  • p21-Activated Kinases / chemistry
  • p21-Activated Kinases / metabolism

Substances

  • Histones
  • Tumor Suppressor Proteins
  • Histone Acetyltransferases
  • KAT7 protein, human
  • PAK1 protein, human
  • p21-Activated Kinases