Lamivudine resistance mutations in patients infected with hepatitis B virus genotype D

World J Gastroenterol. 2011 Dec 7;17(45):4987-92. doi: 10.3748/wjg.v17.i45.4987.

Abstract

Aim: To determine the distribution of viral genotypes for primary or acquired lamivudine resistance.

Methods: A total of 283 patients with chronic hepatitis B virus (HBV) infection (245 patients with chronic hepatitis B and 38 inactive hepatitis B surface antigen carriers) were included in the study. The HBV genotype was determined by using quantitative real-time polymerase chain reaction and sequence analysis, and tyrosine-methionine-aspartate-aspartate (YMDD) motif mutations were determined using the reverse transcriptase hybridization method.

Results: Lamivudine resistance was determined in a total of 25 (10.7%) chronic hepatitis B patients. Eight subjects (4%) had primary resistance to lamivudine, and 17 (53.1%) had secondary resistance to lamivudine. Genotype D, which was isolated from 267 of the patients with chronic HBV infection, was the dominant genotype in Turkey.

Conclusion: Identification of YMDD motif mutations should have a positive impact on the selection of proper antiviral medication for patients, even for those who are nucleoside naïve.

Keywords: Genotype; Hepatitis B virus; Lamivudine; Resistance; Tyrosine-methionine-aspartate-aspartate mutation.

Publication types

  • Multicenter Study

MeSH terms

  • Adult
  • Aged
  • Drug Resistance, Viral / genetics*
  • Female
  • Genotype
  • Hepatitis B virus / drug effects
  • Hepatitis B virus / genetics*
  • Hepatitis B, Chronic / drug therapy*
  • Hepatitis B, Chronic / genetics*
  • Humans
  • Lamivudine / pharmacology
  • Lamivudine / therapeutic use*
  • Male
  • Middle Aged
  • Mutation*
  • Real-Time Polymerase Chain Reaction
  • Reverse Transcriptase Inhibitors / pharmacology
  • Reverse Transcriptase Inhibitors / therapeutic use*
  • Young Adult

Substances

  • Reverse Transcriptase Inhibitors
  • Lamivudine