Validated LC-MS/MS assay for the quantitative determination of clematichinenoside AR in rat plasma and its application to a pharmacokinetic study

Biomed Chromatogr. 2012 Oct;26(10):1282-5. doi: 10.1002/bmc.2691. Epub 2012 Feb 16.

Abstract

This study aimed to develop and validate a liquid chromatography tandem mass spectrometry method for measuring clematichinenoside AR in rat plasma. Clematichinenoside AR was extracted by solid-phase extraction and chromatographed on an XTerra MS C(8) column. Pulchinenoside B4 was used as the internal standard. Elution was achieved using an isocratic mobile phase of acetonitrile with 0.1% acetic acid (21:79, v/v) at a flow-rate of 0.2 mL/min. The detection was performed by multiple reaction monitoring mode via a negative electrospray ionization interface. Standard curves were linear, ranging from 2.5 to 500 ng/mL. The intra- and inter-day precision values were <14.0% and the accuracy was within ±13%. Extraction recovery ranged from 93.2 to 93.9%. This proposed method was successfully applied to a pharmacokinetic study on clematichinenoside AR in rats after oral administration.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Chromatography, Liquid / methods*
  • Chromatography, Liquid / standards
  • Drug Stability
  • Linear Models
  • Oleanolic Acid / analogs & derivatives*
  • Oleanolic Acid / blood
  • Oleanolic Acid / chemistry
  • Oleanolic Acid / pharmacokinetics
  • Rats
  • Reproducibility of Results
  • Saponins / blood*
  • Saponins / chemistry
  • Saponins / pharmacokinetics
  • Sensitivity and Specificity
  • Tandem Mass Spectrometry / methods*
  • Tandem Mass Spectrometry / standards

Substances

  • Saponins
  • clematichinenoside AR2
  • Oleanolic Acid