Polyphosphate: an ancient molecule that links platelets, coagulation, and inflammation

Blood. 2012 Jun 21;119(25):5972-9. doi: 10.1182/blood-2012-03-306605. Epub 2012 Apr 19.

Abstract

Inorganic polyphosphate is widespread in biology and exhibits striking prohemostatic, prothrombotic, and proinflammatory effects in vivo. Long-chain polyphosphate (of the size present in infectious microorganisms) is a potent, natural pathophysiologic activator of the contact pathway of blood clotting. Medium-chain polyphosphate (of the size secreted from activated human platelets) accelerates factor V activation, completely abrogates the anticoagulant function of tissue factor pathway inhibitor, enhances fibrin clot structure, and greatly accelerates factor XI activation by thrombin. Polyphosphate may have utility as a hemostatic agent, whereas antagonists of polyphosphate may function as novel antithrombotic/anti-inflammatory agents. The detailed molecular mechanisms by which polyphosphate modulates blood clotting reactions remain to be elucidated.

Publication types

  • Research Support, N.I.H., Extramural
  • Review

MeSH terms

  • Animals
  • Blood Coagulation / drug effects*
  • Blood Coagulation / physiology
  • Blood Platelets / drug effects*
  • Blood Platelets / metabolism
  • Blood Platelets / physiology
  • Fibrin / metabolism
  • Hemostasis / drug effects
  • Humans
  • Inflammation / blood
  • Inflammation / etiology*
  • Inflammation / metabolism
  • Models, Biological
  • Platelet Adhesiveness / drug effects
  • Platelet Adhesiveness / physiology
  • Polyphosphates / chemistry
  • Polyphosphates / metabolism
  • Polyphosphates / pharmacology*
  • Signal Transduction / drug effects
  • Signal Transduction / physiology
  • Thrombin / metabolism

Substances

  • Polyphosphates
  • Fibrin
  • Thrombin